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Compounds

Cat No. Product Name
T10876 CPA inhibitor Carboxypeptidase inhibitor Carboxypeptidase
CPA inhibitor 是一种有效的羧肽酶 A (CPA) 抑制剂,Ki 值为 0.32 μM。
T1804 HPGDS inhibitor 1 HPGDS-inhibitor-1 PGE Synthase
HPGDS inhibitor 1 是口服具有活性的HPGDS 选择性抑制剂,在酶和细胞分析中的IC50值分别为 0.6 nM 和 32 nM,但对 L-PGDS、mPGES、COX-1、COX-2 、5-LOX 无抑制作用。
T8766 GOT1 inhibitor-1 GOT1 inhibitor 2c Others
GOT1 inhibitor-1 是一种新型的、非共价的谷氨酸草酰乙酸转氨酶 1 (GOT1) 抑制剂(IC50:8.2 uM),是一种戊酸衍生物。 它可用于以及胰腺导管腺癌 (PDAC) 。
T5451 Eph inhibitor 2 Ehp-inhibitor-1 Ephrin Receptor
Ehp-inhibitor-1 是一种 Eph 家族酪氨酸激酶抑制剂。
T4338 USP7/USP47 inhibitor USP7/47 inhibitor-1 DUB
USP7/USP47 inhibitor 是一种选择性泛素特异性蛋白酶 7/47 抑制剂,EC50值分别为 0.42 μM 和 1.0 μM。
T3593 Src Inhibitor 1 Src Kinase Inhibitor 1,Src-l1 Src
Src Inhibitor 1 是一种选择性的、高效的、ATP-竞争性的双位点 Src 酪氨酸激酶抑制剂,能够抑制 Src (IC50:44 nM) 和 Lck (IC50:88 nM)。
T6335 Tie2 kinase inhibitor 1 Tie2 kinase inhibitor Tie-2
Tie2 kinase inhibitor 1 是Tie2激酶选择性抑制剂9IC50:250 nM),具有抗癌作用。
T38683 SCD1 inhibitor-3 SCD1-IN-3,SCD1 inhibitor 17a Dehydrogenase
SCD1 inhibitor-3 is a highly effective and orally available compound that inhibits SCD1 with remarkable safety. It demon...
T2350 MALT1 inhibitor MI-2 MI 2 (MALT1 inhibitor),MALT1 inhibitor,MI 2 MALT
MI 2 (MALT1 inhibitor) 是一种MALT1抑制剂 (IC50=5.84 μM),对动物无毒性。它能够直接与 MALT1 结合,不可逆地抑制蛋白酶功能,并伴有 NF-κB 报告子活性抑制、c-REL 核定位抑制和 NF-κ...
T5817 PKC-theta inhibitor hcl PKC-theta inhibitor PKC
PKC-theta inhibitor 是一种选择性 PKC-θ 抑制剂 (IC50:12 nM)。
T5524 Aurora kinase inhibitor-3 Aurora Kinase Inhibitor III Aurora Kinase
Aurora kinase inhibitor-3 是一种有效的,选择性 Aurora A 激酶抑制剂,IC50为 42 nM。
T24141 HIV-1 Inhibitor 18A HIV-1 Inhibitor-18A HIV Protease
HIV-1 Inhibitor 18A 特异性抑制多种 HIV-1 分离株的进入。
T4191 Multi-kinase inhibitor 1 Multi-kinase inhibitor I Others , PDGFR , Bcr-Abl , c-Kit
Multi-kinase inhibitor 1 是多激酶抑制剂。它有用于导致与酪氨酸激酶活性异常或失控有关的疾病或失调的潜力,特别是与c-Kit,PDGF-R,Bcr-abl 活性相关的疾病。
T3189 B7/CD28 interaction inhibitor 1 CTLA-4 inhibitor Others
CTLA-4 inhibitor 是B7.1-CD28相互作用抑制剂(IC50:50 nM)。
T12348 P38α inhibitor 1 ARRY-797,P38a inhibitor 1,P38alpha inhibitor 1 p38 MAPK
p38α inhibitor 1是p38α的抑制剂。
T4167 Raf inhibitor 1 dihydrochloride B-Raf inhibitor 1 dihydrochloride Raf
B-Raf inhibitor 1 dihydrochloride 是 Raf 激酶抑制剂,对 B-RafWT、B-RafV600E 和 C-Raf 的Ki 分别为 1、1 和 0.3 nM。
T10678 Carboxypeptidase G2 (CPG2) Inhibitor Carboxypeptidase G2 Inhibitor,CPG2 Inhibitor Carboxypeptidase
Carboxypeptidase G2 (CPG2) Inhibitor 是新型的羧肽酶 G2(CPG2)抑制剂,显示出抗癌活性。
T9040 Aurora kinase inhibitor-2 Aurora Kinase Inhibitor II,IUN-70219 Aurora Kinase
Aurora kinase inhibitor-2 是一种可渗透细胞的苯胺喹唑啉,可抑制极光激酶的活性,对Aurora A 和Aurora B 的IC50分别为 390 nM 和 240 nM。
T2457 IRAK-1-4 Inhibitor I IRAK-1/4 Inhibitor,IRAK-1/4 Inhibitor I IRAK
IRAK-1/4 Inhibitor 是一种IRAK1/4双重抑制剂,其IC50分别为 0.2 μM 和 0.3 μM。
T35827L PKCε Inhibitor Peptide acetate PKCε Inhibitor Peptide acetate(182683-50-7 Free base) PKC
PKCε Inhibitor Peptide acetate 是一种特异性 PKCε 抑制剂,含有其特定受体活化 C 激酶 (RACK) 的位点。 PKCε Inhibitor Peptide acetate 抑制 PKCε 的转运,但不抑...
CPA inhibitor
T10876
synonym: Carboxypeptidase inhibitor
Target:
HPGDS inhibitor 1
T1804
synonym: HPGDS-inhibitor-1
Target:
GOT1 inhibitor-1
T8766
synonym: GOT1 inhibitor 2c
Target:
Eph inhibitor 2
T5451
synonym: Ehp-inhibitor-1
Target:
USP7/USP47 inhibitor
T4338
synonym: USP7/47 inhibitor-1
Target:
Src Inhibitor 1
T3593
synonym: Src Kinase Inhibitor 1,Src-l1
Target:
Tie2 kinase inhibitor 1
T6335
synonym: Tie2 kinase inhibitor
Target:
SCD1 inhibitor-3
T38683
synonym: SCD1-IN-3,SCD1 inhibitor 17a
Target:
MALT1 inhibitor MI-2
T2350
synonym: MI 2 (MALT1 inhibitor),MALT1 inhibitor,MI 2
Target:
PKC-theta inhibitor hcl
T5817
synonym: PKC-theta inhibitor
Target:
Aurora kinase inhibitor-3
T5524
synonym: Aurora Kinase Inhibitor III
Target:
HIV-1 Inhibitor 18A
T24141
synonym: HIV-1 Inhibitor-18A
Target:
Multi-kinase inhibitor 1
T4191
synonym: Multi-kinase inhibitor I
Target:
B7/CD28 interaction inhibitor 1
T3189
synonym: CTLA-4 inhibitor
Target:
p38α inhibitor 1
T12348
synonym: ARRY-797,P38a inhibitor 1,P38alpha inhibitor 1
Target:
Raf inhibitor 1 dihydrochloride
T4167
synonym: B-Raf inhibitor 1 dihydrochloride
Target:
Carboxypeptidase G2 (CPG2) Inhibitor
T10678
synonym: Carboxypeptidase G2 Inhibitor,CPG2 Inhibitor
Target:
Aurora kinase inhibitor-2
T9040
synonym: Aurora Kinase Inhibitor II,IUN-70219
Target:
IRAK-1-4 Inhibitor I
T2457
synonym: IRAK-1/4 Inhibitor,IRAK-1/4 Inhibitor I
Target:
PKCε Inhibitor Peptide acetate
T35827L
synonym: PKCε Inhibitor Peptide acetate(182683-50-7 Free base)
Target:
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