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MLT-943

Name: MLT-943
Brand: TargetMol
SKU: T9216
Price: 74 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T9216Cas No. 1832576-04-1

Alias MLT943

MLT-943 is a potent, selective, and orally active MALT1 protease inhibitor [1].

MLT-943

🥰Excellent

Purity: 99.82%

Catalog No. T9216Alias MLT943Cas No. 1832576-04-1

MLT-943 is a potent, selective, and orally active MALT1 protease inhibitor [1].

Pack Size	Price	Availability
1 mg	$74	In Stock
5 mg	$158	In Stock
10 mg	$238	In Stock
25 mg	$398	In Stock
50 mg	$567	In Stock
100 mg	$768	In Stock
200 mg	$987	In Stock
1 mL x 10 mM (in DMSO)	$173	In Stock

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Batch Information

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Purity:99.82%

Resource Download

COA HPLC HNMR

Product Introduction

Bioactivity

Description	MLT-943 is a potent, selective, and orally active MALT1 protease inhibitor [1].
In vitro	MLT-943 inhibits stimulated-IL-2 secretion in PBMC or in whole blood with a similar?IC50?across species (0.07-0.09 μM in PBMC, 0.6-0.8 μM in whole blood).
Synonyms	MLT943

Chemical Properties

Molecular Weight	414.77
Formula	C₁₆H₁₄ClF₃N₆O₂
Cas No.	1832576-04-1
Smiles	CO[C@@H](C)c1c(NC(=O)Nc2ccnc(c2)C(F)(F)F)cnc2cc(Cl)nn12
Relative Density.	1.56 g/cm3 (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 247 mg/mL (595.51 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.4110 mL	12.0549 mL	24.1097 mL	120.5487 mL
5 mM	0.4822 mL	2.4110 mL	4.8219 mL	24.1097 mL
10 mM	0.2411 mL	1.2055 mL	2.4110 mL	12.0549 mL
20 mM	0.1205 mL	0.6027 mL	1.2055 mL	6.0274 mL
50 mM	0.0482 mL	0.2411 mL	0.4822 mL	2.4110 mL
100 mM	0.0241 mL	0.1205 mL	0.2411 mL	1.2055 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc