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TargetMol | Tags GPCR/G Protein
TargetMol | Tags Neuroscience

Neuropeptide Y Receptor

Neuropeptide Y receptors are a family of receptors belonging to class A G-protein coupled receptors and they are activated by the closely related peptide hormones neuropeptide Y, peptide YY and pancreatic polypeptide. These receptors are involved in the control of a diverse set of behavioral processes including appetite, circadian rhythm, and anxiety.

Pancreatic Polypeptide, rat acetate
TP1044L
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.
  • $238
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Selvigaltin
T637511978336-95-6In house
Selvigaltin (GB1211) is a Gal-3 inhibitor with potential anticancer activity. Selvigaltin is used in the study of cirrhosis and cancer.
  • $289
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Peptide YY (PYY) (3-36), human
TP1059126339-09-1
Peptide YY (PYY) (3-36), human (Peptide YY (3-36)), is a gut hormone peptide that acts as a Y2 receptor agonist to reduce appetite.
  • $76
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BIBO3304 TFA
T10539191868-14-1
BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 receptor).
  • $98
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BWX 46 Acetate
T21611L
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.
  • $253
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DF-1012 FA
T27158L In house
DF-1012 FA is a structural analog of DF-1012, a neuropeptide inhibitor used in the study of asthma and cough.
  • $195 TargetMol
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NPY 5RA972
T23087439861-56-0
neuropeptide Y Y5 receptor antagonist
  • $39
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[Leu31,Pro34]-Neuropeptide Y (porcine)
TP2206125580-28-1
High affinity neuropeptide Y Y1 receptor agonist
  • $58
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Galantide acetate
T15368L
Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P. Galantide acetate recognizes two classes of galanin binding sites (KD<0.1 nM and ~6 nM) in the rat hypothalamus. Galantide acetate dose dependently (IC50=1.0 nM) antagonizes the galanin-mediated inhibition of the glucose-induced insulin secretion from mouse pancreatic islets. Galantide acetate appears to bind to a single population of SP receptors (KD~40 nM).
  • $158 TargetMol
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RFRP3(human) acetate(311309-27-0 free base)
TP1936L1
RFRP-3(human) acetate, a human GnIH peptide homolog, is a potent inhibitor of gonadotropin secretion by inhibiting Ca2+ mobilization. RFRP-3(human) acetate is a NPFF1 receptor agonist, it inhibits forskolin-induced production of cAMP with an IC50 of 0.7 n
  • $80
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ML 154
T229941345964-89-7
neuropeptide S receptor (NPSR) antagonist
  • $53
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ntncb hydrochloride
T23094191931-56-3
NTNCB hydrochloride is an antagonist of neuropeptide Y (NPY) Y5 receptor.
  • $45
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Velneperit
T17222342577-38-2
Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.
  • $31
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Galanin Receptor Ligand M35 TFA
TP1704
Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of the galanin receptor (Kd = 0.1 nM).
  • $113
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RF9 acetate
T16738L
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.
  • $59
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Neuropeptide S (Mouse) acetate
TP1981L
Neuropeptide S (Mouse) acetate is a bioactive peptide. Neuropeptide S (Mouse) acetate, as a neurotransmitter neuromodulator of 20 amino acids, can be used for the research of arousal, anxiety, locomotion, feeding behaviors, memory and drug addiction[1].
  • $148
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Spexin acetate(1370290-58-6 free base)
TP1930L1
Spexin acetate is a potent galanin receptor 2 3 (GAL2 GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galanin receptor 1. Endogenous satiety-inducing peptide; inhibits long chain fatty acid uptake by ad
  • $116
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Galanin (1-16), mouse, porcine, rat
TP1380125118-77-6
Galanin (1-16), mouse, porcine, rat, is a hippocampal galanin receptor agonist (Kd = 3 nM) exhibiting high biological activity on locus coeruleus neurons.
  • $167
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Neuropeptide S (Rat) acetate
TP1982L
Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now named NPS receptor. Neuropeptide S (Rat) acetate can be used for the research of nervous system disease [1].
  • $148
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Neuropeptide FF acetate(99566-27-5 free base)
TP1074L
Neuropeptide FF acetate(99566-27-5 free base) (NPFF acetate) is an octapeptide belonging to the RF amide family. NPFF interacts with G-protein-coupled receptors NPFF (1) and NPFF (2).
  • $147
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CYM2503
T89631308833-36-4
CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. It has no affinity for the orthosteric galanin binding site of the receptor (as measured by its inability to displace iodinated galanin, or to induce IP1 accumulation on its own).
  • $31
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JNJ-31020028
T19971094873-14-9
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22, rat); it exhibits >100-fold selectivity for Y2 versus human Y1 Y4 Y5 receptors.
  • $43
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BMS-193885
T14671186185-03-5
BMS-193885 is a selective, brain-penetrant, and competitive antagonist of the neuropeptide Y1 receptor with a Ki of 3.3 nM, and an IC50 of 5.9 nM for hY1.
  • $29
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MK-0557
TQ0286328232-95-7
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).
  • $30
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