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GSK-2881078 (Alias: GSK2881078, GSK 2881078)

Name: GSK-2881078
Brand: TargetMol
SKU: T3618
Price: 38 USD
Availability: InStock
Rating: 5 (10 reviews)

Catalog No. T3618 Copy Product Info

Purity: 98.81%

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GSK-2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting to improve their physical function.

GSK-2881078

Copy Product Info

🥰Excellent

Catalog No. T3618

Alias GSK2881078, GSK 2881078

GSK-2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting to improve their physical function.

Cas No. 1539314-06-1

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Pack Size	Price	USA Stock	Global Stock
5 mg	$38	In Stock	In Stock
10 mg	$58	In Stock	In Stock
25 mg	$128	In Stock	In Stock
50 mg	$208	In Stock	In Stock
100 mg	$347	In Stock	In Stock
200 mg	$497	-	In Stock
1 mL x 10 mM (in DMSO)	$42	In Stock	In Stock

In stock · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)

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For research use only—not for human use. No sales to individuals. Use as intended only.

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Purity:98.81%

Color:White

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	GSK-2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting to improve their physical function.
Synonyms	GSK2881078, GSK 2881078

Chemical Properties

Molecular Weight	330.33
Formula	C₁₄H₁₃F₃N₂O₂S
Cas No.	1539314-06-1
Smiles	C[C@H](CS(C)(=O)=O)n1ccc2c(c(ccc12)C#N)C(F)(F)F
Relative Density.	1.36 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 60 mg/mL (181.64 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.0273 mL	15.1364 mL	30.2728 mL	151.3638 mL
5 mM	0.6055 mL	3.0273 mL	6.0546 mL	30.2728 mL
10 mM	0.3027 mL	1.5136 mL	3.0273 mL	15.1364 mL
20 mM	0.1514 mL	0.7568 mL	1.5136 mL	7.5682 mL
50 mM	0.0605 mL	0.3027 mL	0.6055 mL	3.0273 mL
100 mM	0.0303 mL	0.1514 mL	0.3027 mL	1.5136 mL

Note : The dilution table applies only to solid products. For liquid products, please calculate the stock solution based on the stated concentration and/or density.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc