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PKI-166 hydrochloride

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Catalog No. T36643Cas No. 2230253-82-2

Potent EGFR-kinase inhibitor (IC50 = 0.7 nM). Displays >3000-fold selectivity against a panel of serine/threonine kinases. Reduces metastasis and angiogenesis in a mouse model of pancreatic cancer. Antihypertensive and orally bioavailable.

PKI-166 hydrochloride
Other Forms of PKI-166 hydrochloride:
PKI-166T16549187724-61-4
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PKI-166 hydrochloride

😃Good
Catalog No. T36643Cas No. 2230253-82-2
Potent EGFR-kinase inhibitor (IC50 = 0.7 nM). Displays >3000-fold selectivity against a panel of serine/threonine kinases. Reduces metastasis and angiogenesis in a mouse model of pancreatic cancer. Antihypertensive and orally bioavailable.
Pack SizePriceAvailabilityQuantity
10 mgTBD35 days
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Product Introduction

Bioactivity
Description
Potent EGFR-kinase inhibitor (IC50 = 0.7 nM). Displays >3000-fold selectivity against a panel of serine/threonine kinases. Reduces metastasis and angiogenesis in a mouse model of pancreatic cancer. Antihypertensive and orally bioavailable.
Targets&IC50
EGFR tyrosine kinase:0.7 nM (IC50)
Chemical Properties
Molecular Weight366.85
FormulaC20H19ClN4O
Cas No.2230253-82-2
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.
Solubility Information
DMSO: Soluble

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Keywords

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