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Gabazine

Name: Gabazine
Brand: TargetMol
SKU: T7622
Price: 47 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T7622Cas No. 104104-50-9

Alias SR95531

Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)

Gabazine

🥰Excellent

Purity: 99.24%

Catalog No. T7622Alias SR95531Cas No. 104104-50-9

Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)

Pack Size	Price	Availability
5 mg	$47	In Stock
10 mg	$72	In Stock
25 mg	$143	In Stock
50 mg	$272	In Stock
100 mg	$488	In Stock
200 mg	$659	In Stock
1 mL x 10 mM (in DMSO)	$52	In Stock

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Batch Information

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Purity:99.24%

Resource Download

COA LCMS HNMR LCMS

Product Introduction

Bioactivity

Description	Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)
Targets&IC50	GABAA:74-150 nM(ki)
In vivo	Gabazine is effective against GABAA receptor isoforms from mice, rats, and humans[1].
Synonyms	SR95531

Chemical Properties

Molecular Weight	368.23
Formula	C₁₅H₁₈BrN₃O₃
Cas No.	104104-50-9
Smiles	Br.COc1ccc(cc1)-c1ccc(=N)n(CCCC(O)=O)n1
Relative Density.	no data available
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 75 mg/mL (203.68 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.7157 mL	13.5785 mL	27.1569 mL	135.7847 mL
5 mM	0.5431 mL	2.7157 mL	5.4314 mL	27.1569 mL
10 mM	0.2716 mL	1.3578 mL	2.7157 mL	13.5785 mL
20 mM	0.1358 mL	0.6789 mL	1.3578 mL	6.7892 mL
50 mM	0.0543 mL	0.2716 mL	0.5431 mL	2.7157 mL
100 mM	0.0272 mL	0.1358 mL	0.2716 mL	1.3578 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc