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H2L 5765834

Name: H2L 5765834
Brand: TargetMol
SKU: T22834
Price: 56 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T22834Cas No. 420841-84-5

H2L 5765834 is a lysophosphatidic acid receptors antagonist

H2L 5765834

🥰Excellent

Purity: 99.47%

Catalog No. T22834Cas No. 420841-84-5

H2L 5765834 is a lysophosphatidic acid receptors antagonist

Pack Size	Price	Availability
1 mg	$56	In Stock
5 mg	$122	In Stock
10 mg	$197	In Stock
25 mg	$372	In Stock
50 mg	$553	In Stock
100 mg	$787	In Stock
1 mL x 10 mM (in DMSO)	$133	In Stock

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Batch Information

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Purity:99.47%

Resource Download

COA HPLC HNMR

Product Introduction

Bioactivity

Description	H2L 5765834 is a lysophosphatidic acid receptors antagonist
Targets&IC50	LPA3 receptor:752 nM (IC50), LPA5 receptor:463 nM (IC50), LPA1 receptor:94 nM (IC50)

Chemical Properties

Molecular Weight	404.33
Formula	C₂₁H₁₂N₂O₇
Cas No.	420841-84-5
Smiles	OC(=O)c1ccc2C(=O)N(C(=O)c2c1)c1cccc(Oc2ccc(cc2)[N+]([O-])=O)c1
Relative Density.	1.544 g/cm3 (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 55 mg/mL (136.03 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.4732 mL	12.3661 mL	24.7323 mL	123.6614 mL
5 mM	0.4946 mL	2.4732 mL	4.9465 mL	24.7323 mL
10 mM	0.2473 mL	1.2366 mL	2.4732 mL	12.3661 mL
20 mM	0.1237 mL	0.6183 mL	1.2366 mL	6.1831 mL
50 mM	0.0495 mL	0.2473 mL	0.4946 mL	2.4732 mL
100 mM	0.0247 mL	0.1237 mL	0.2473 mL	1.2366 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc