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Tyrphostin A25

Name: Tyrphostin A25
Brand: TargetMol
SKU: T21622
Price: 33 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T21622Cas No. 118409-58-8

Alias Tyrphostin AG 82, RG-50875, AG-82

Tyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist with an IC50 value of 0.94 μM for GPR35 and an EC50 value of 5.3 μM for GPR35.

Tyrphostin A25

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Purity: 98.76%

Catalog No. T21622Alias Tyrphostin AG 82, RG-50875, AG-82Cas No. 118409-58-8

Tyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist with an IC50 value of 0.94 μM for GPR35 and an EC50 value of 5.3 μM for GPR35.

Pack Size	Price	Availability
2 mg	$33	In Stock
5 mg	$52	In Stock
10 mg	$75	In Stock
25 mg	$123	In Stock
50 mg	$182	In Stock
100 mg	$269	In Stock

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Purity:98.76%

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COA HNMR HPLC

Product Introduction

Bioactivity

Description	Tyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist with an IC50 value of 0.94 μM for GPR35 and an EC50 value of 5.3 μM for GPR35.
Targets&IC50	GPR35:5.3 µM, GPR35:0.94 µM
In vitro	In the human epidermoid carcinoma cell line A431, Tyrphostin A25 inhibited the activity of epidermal growth factor receptor kinase with an IC50 value of 3 μM.[1]
Synonyms	Tyrphostin AG 82, RG-50875, AG-82

Chemical Properties

Molecular Weight	202.17
Formula	C₁₀H₆N₂O₃
Cas No.	118409-58-8
Smiles	C(=C(C#N)C#N)C1=CC(O)=C(O)C(O)=C1
Relative Density.	1.569 g/cm3

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Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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