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σ1 Receptor antagonist-1

Name: σ1 Receptor antagonist-1
Brand: TargetMol
SKU: T9244
Price: 35 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T9244Cas No. 1204401-49-9

σ1 Receptor antagonist-1 is a selective σ1 receptor antagonist.

σ1 Receptor antagonist-1

🥰Excellent

Purity: 99.8%

Catalog No. T9244Cas No. 1204401-49-9

σ1 Receptor antagonist-1 is a selective σ1 receptor antagonist.

Pack Size	Price	Availability
5 mg	$35	In Stock
10 mg	$56	In Stock
25 mg	$121	In Stock
50 mg	$198	In Stock
100 mg	$288	In Stock
200 mg	$413	In Stock
1 mL x 10 mM (in DMSO)	$38	In Stock

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Batch Information

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Purity:99.8%

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description	σ1 Receptor antagonist-1 is a selective σ1 receptor antagonist.
In vitro	σ1 Receptor antagonist-1 (compound 9) (10 μM; 48 hours) arrests cell cycle at G0/G1 phase to inhibit cell growth, and induces?apoptosis?of MCF-7/ADR cells[1]

Chemical Properties

Molecular Weight	337.48
Formula	C₂₁H₂₃NOS
Cas No.	1204401-49-9
Smiles	O=C1CC(Sc2ccccc12)C1CCN(Cc2ccccc2)CC1
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 90 mg/mL (266.68 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.9631 mL	14.8157 mL	29.6314 mL	148.1569 mL
5 mM	0.5926 mL	2.9631 mL	5.9263 mL	29.6314 mL
10 mM	0.2963 mL	1.4816 mL	2.9631 mL	14.8157 mL
20 mM	0.1482 mL	0.7408 mL	1.4816 mL	7.4078 mL
50 mM	0.0593 mL	0.2963 mL	0.5926 mL	2.9631 mL
100 mM	0.0296 mL	0.1482 mL	0.2963 mL	1.4816 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc