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Khellin

Name: Khellin
Brand: TargetMol
SKU: T1431
Rating: 4.5 (1 reviews)

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Catalog No. T1431Cas No. 82-02-0

Alias Visammin, Methafrone, Amicardine

Khellin (Methafrone) is a vasodilator that also has bronchodilatory action.

Khellin

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Purity: 99.95%

Catalog No. T1431Alias Visammin, Methafrone, AmicardineCas No. 82-02-0

Khellin (Methafrone) is a vasodilator that also has bronchodilatory action.

Pack Size	Price	EUR Warehouse	Global Warehouse
10 mg	$31	Backorder	Backorder
25 mg	$47	Backorder	Backorder
50 mg	$68	Backorder	Backorder
100 mg	$89	Backorder	Backorder
500 mg	$219	Backorder	Backorder
1 mL x 10 mM (in DMSO)	$29	Backorder	Backorder

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Expected start date of shipmentEUR Warehouse [1-2 days] Global Warehouse [5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

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Purity:99.95%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	Khellin (Methafrone) is a vasodilator that also has bronchodilatory action.
Targets&IC50	EGFR:0.15 µM (IC50)
Synonyms	Visammin, Methafrone, Amicardine

Chemical Properties

Molecular Weight	260.24
Formula	C₁₄H₁₂O₅
Cas No.	82-02-0
Smiles	COc1c2ccoc2c(OC)c2oc(C)cc(=O)c12
Relative Density.	1.301 g/cm3

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 12 mg/mL (46.11 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.8426 mL	19.2130 mL	38.4261 mL	192.1303 mL
5 mM	0.7685 mL	3.8426 mL	7.6852 mL	38.4261 mL
10 mM	0.3843 mL	1.9213 mL	3.8426 mL	19.2130 mL
20 mM	0.1921 mL	0.9607 mL	1.9213 mL	9.6065 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc