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Labetalone hydrochloride

Name: Labetalone hydrochloride
Brand: TargetMol
SKU: T35326
Price: 29 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T35326Cas No. 96441-14-4

Alias Labetalone hydrochloride, Benzoic amide

Labetalone hydrochloride is an orally effective adrenergic receptor blocking drug that competitively antagonizes both α and β receptor sites.

Labetalone hydrochloride

🥰Excellent

Purity: 99.58%

Catalog No. T35326Alias Labetalone hydrochloride, Benzoic amideCas No. 96441-14-4

Labetalone hydrochloride is an orally effective adrenergic receptor blocking drug that competitively antagonizes both α and β receptor sites.

Pack Size	Price	Availability
25 mg	$38	In Stock
50 mg	$59	In Stock
100 mg	$98	In Stock
200 mg	$153	In Stock
500 mg	$260	In Stock
1 mL x 10 mM (in DMSO)	$29	In Stock

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Purity:99.58%

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COA HNMR LCMS

Product Introduction

Bioactivity

Description	Labetalone hydrochloride is an orally effective adrenergic receptor blocking drug that competitively antagonizes both α and β receptor sites.
Synonyms	Labetalone hydrochloride, Benzoic amide

Chemical Properties

Molecular Weight	362.85
Formula	C₁₉H₂₃ClN₂O₃
Cas No.	96441-14-4
Smiles	Cl.CC(CCc1ccccc1)NCC(=O)c1ccc(O)c(c1)C(N)=O

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 27.5 mg/mL (75.79 mM), Sonication is recommended.

In Vivo Formulation

10% DMSO+40% PEG300+5% Tween 80+45% Saline: 2 mg/mL (5.51 mM), Sonication is recommended.

Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.7560 mL	13.7798 mL	27.5596 mL	137.7980 mL
5 mM	0.5512 mL	2.7560 mL	5.5119 mL	27.5596 mL
10 mM	0.2756 mL	1.3780 mL	2.7560 mL	13.7798 mL
20 mM	0.1378 mL	0.6890 mL	1.3780 mL	6.8899 mL
50 mM	0.0551 mL	0.2756 mL	0.5512 mL	2.7560 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc