Powder: -20°C for 3 years | In solvent: -80°C for 1 year
EZH2-IN-5 is a highly effective inhibitor of EZH2, displaying remarkable potency against both wild-type and mutant Tyr641 EZH2, with IC50 values of 1.52 nM and 4.07 nM, respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | Inquiry | $ 970.00 |
Description | EZH2-IN-5 is a highly effective inhibitor of EZH2, displaying remarkable potency against both wild-type and mutant Tyr641 EZH2, with IC50 values of 1.52 nM and 4.07 nM, respectively. |
Targets&IC50 | EZH2 (Y641F):4.07 nM (IC50), EZH2 (WT):1.52 nM (IC50) |
In vitro | EZH2-IN-5 (compound 276) effectively suppresses the proliferation of WSUDLCL2 cell lines, demonstrating an inhibitory concentration (IC50) of 187.28 nM[1]. |
Synonyms | EZH2-IN-5 |
Molecular Weight | 517.512 |
Formula | C26H37BrN4O2 |
CAS No. | 1403258-69-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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EZH2-IN-5 1403258-69-4 EZH2 IN 5 EZH-2-IN-5 EZH2IN5 inhibitor inhibit