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A 410099.1

Name: A 410099.1
Brand: TargetMol
SKU: T36890
Price: 149 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T36890Cas No. 762274-58-8

Alias A410099.1

A410099.1 is a BIRC (baculoviral IAP repeat-containing protein) inhibitor with EC50 values of 4.6, 9.2, 15.6, 19.9, and 93.9 nM for BIRC2/3/4/7/8 respectively, suitable for studying E3 ligases and PROTAC synthesis.

A 410099.1

🥰Excellent

Purity: 99.30%

Catalog No. T36890Alias A410099.1Cas No. 762274-58-8

Pack Size	Price	USA Warehouse	Global Warehouse	Quantity
1 mg	$149	-	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

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Purity:99.30%

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COA

Product Introduction

Bioactivity

Description	A410099.1 is a BIRC (baculoviral IAP repeat-containing protein) inhibitor with EC50 values of 4.6, 9.2, 15.6, 19.9, and 93.9 nM for BIRC2/3/4/7/8 respectively, suitable for studying E3 ligases and PROTAC synthesis.
Targets&IC50	BIRC8:93.9 nM (EC50), BIRC4:15.6 nM ( EC50), BIRC3:9.2 nM (EC50), BIRC7:19.9 nM (EC50), BIRC2:4.6 nM (EC50)
Synonyms	A410099.1

Chemical Properties

Molecular Weight	505.1
Formula	C₂₇H₄₁ClN₄O₃
Cas No.	762274-58-8
Smiles	Cl.CN[C@@H](C)C(=O)N[C@@H](C1CCCCC1)C(=O)N1CCC[C@H]1C(=O)N[C@@H]1CCCc2ccccc12 \|@:9\|
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 40 mg/mL (79.19 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.9798 mL	9.8990 mL	19.7981 mL	98.9903 mL
5 mM	0.3960 mL	1.9798 mL	3.9596 mL	19.7981 mL
10 mM	0.1980 mL	0.9899 mL	1.9798 mL	9.8990 mL
20 mM	0.0990 mL	0.4950 mL	0.9899 mL	4.9495 mL
50 mM	0.0396 mL	0.1980 mL	0.3960 mL	1.9798 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc