Shopping Cart

Your shopping cart is currently empty

Didesethyl chloroquine

Name: Didesethyl chloroquine
Brand: TargetMol
SKU: T11039
Price: 30 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T11039Cas No. 4298-14-0

Alias Bisdesethylchloroquine

Didesethyl chloroquine (Bisdesethylchloroquine) is an effective myocardial inhibitor. Didesethyl chloroquine (Bisdesethylchloroquine) is the main metabolite of the antimalarial drug chloroquine.

Didesethyl chloroquine

🥰Excellent

Purity: 97.91%

Catalog No. T11039Alias BisdesethylchloroquineCas No. 4298-14-0

Didesethyl chloroquine (Bisdesethylchloroquine) is an effective myocardial inhibitor. Didesethyl chloroquine (Bisdesethylchloroquine) is the main metabolite of the antimalarial drug chloroquine.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$53	In Stock	In Stock
5 mg	$133	In Stock	In Stock
10 mg	$197	In Stock	In Stock
25 mg	$331	In Stock	In Stock
50 mg	$472	In Stock	In Stock
1 mL x 10 mM (in DMSO)	$30	In Stock	In Stock

Add to Cart

Add to Quotation

In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

Questions

Batch Information

Select Batch

Purity:97.91%

Resource Download

COA HPLC HNMR

Product Introduction

Bioactivity

Description	Didesethyl chloroquine (Bisdesethylchloroquine) is an effective myocardial inhibitor. Didesethyl chloroquine (Bisdesethylchloroquine) is the main metabolite of the antimalarial drug chloroquine.
Targets&IC50	P. falciparum (HB3):0.0472 μM, P. falciparum (PH3):1.2563 μM, P. falciparum (3D7):0.0553 μM, P. falciparum:58.3 μM, P. falciparum (K1):1.3386 μM
Synonyms	Bisdesethylchloroquine

Chemical Properties

Molecular Weight	263.77
Formula	C₁₄H₁₈ClN₃
Cas No.	4298-14-0
Smiles	CC(CCCN)Nc1ccnc2cc(Cl)ccc12
Relative Density.	1.208g/cm3

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 90 mg/mL (341.21 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.7912 mL	18.9559 mL	37.9118 mL	189.5591 mL
5 mM	0.7582 mL	3.7912 mL	7.5824 mL	37.9118 mL
10 mM	0.3791 mL	1.8956 mL	3.7912 mL	18.9559 mL
20 mM	0.1896 mL	0.9478 mL	1.8956 mL	9.4780 mL
50 mM	0.0758 mL	0.3791 mL	0.7582 mL	3.7912 mL
100 mM	0.0379 mL	0.1896 mL	0.3791 mL	1.8956 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc