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Pirmagrel
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Catalog No. T67958Cas No. 85691-74-3
pirmagrel is a potent thromboxane synthase inhibitor.
Pirmagrel
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Purity: 98.02%
Catalog No. T67958Cas No. 85691-74-3
pirmagrel is a potent thromboxane synthase inhibitor.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $75 | In Stock | In Stock | |
| 5 mg | $179 | In Stock | In Stock | |
| 10 mg | $270 | In Stock | In Stock | |
| 25 mg | $506 | In Stock | In Stock | |
| 50 mg | $680 | In Stock | In Stock | |
| 100 mg | $990 | - | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products.If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
Batch Information
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Purity:98.02%
Appearance:Solid
Color:White
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Product Introduction
Pirmagrel AI Summary
Pirmagrel inhibits thromboxane synthase with an IC50 value of approximately 3.0-3.2 nM in in vitro assays using lysed human platelets as the enzyme source. It also has significant inhibitory activity against Prostaglandin G/H synthase with an IC50 of 10,000 nM. In addition to its effects on enzyme activity, Pirmagrel shows antiviral activity against SARS-CoV-2 by inhibiting the virus-induced cytotoxicity in VERO-6 cells at 10 µM after 48 hours of exposure to a 0.01 MOI SARS-CoV-2 virus, with an IC50 value greater than 19,952.62 nM. The compound's partition coefficient (LogP) is 1.1..
Note: Summary generated by AI. Data source: ChEMBL 
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | pirmagrel is a potent thromboxane synthase inhibitor. |
| Molecular Weight | 232.28 |
| Formula | C13H16N2O2 |
| Cas No. | 85691-74-3 |
| Smiles | C(CCCCC(O)=O)C=1N2C(=CN=C2)C=CC1 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 60 mg/mL (258.31 mM), Sonication is recommended.  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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