Shopping Cart

Your shopping cart is currently empty

DPCPX

Name: DPCPX
Brand: TargetMol
SKU: T22744
Price: 31 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T22744Cas No. 102146-07-6

Alias PD 116948

DPCPX (PD 116948) is an A1 adenosine receptor antagonist

DPCPX

🥰Excellent

Purity: 99.93%

Catalog No. T22744Alias PD 116948Cas No. 102146-07-6

DPCPX (PD 116948) is an A1 adenosine receptor antagonist

Pack Size	Price	USA Warehouse	Global Warehouse
5 mg	$31	In Stock	In Stock
10 mg	$41	In Stock	In Stock
25 mg	$65	In Stock	In Stock
50 mg	$98	In Stock	In Stock
1 mL x 10 mM (in DMSO)	$45	In Stock	In Stock

Add to Cart

Add to Quotation

In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

Select Batch

Purity:99.93%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	DPCPX (PD 116948) is an A1 adenosine receptor antagonist
Targets&IC50	[3H]-CHA binding to A1 receptor (rat whole brain membranes):0.46 nM (Ki), [3H]-NECA binding to A2 receptor (rat striatal membranes):340 nM (Ki)
In vivo	DPCPX, a selective adenosine A1 receptor antagonist, enhances the antidepressant-like effects of imipramine, escitalopram, and reboxetine in mice behavioral tests
Synonyms	PD 116948

Chemical Properties

Molecular Weight	304.39
Formula	C₁₆H₂₄N₄O₂
Cas No.	102146-07-6
Smiles	C(CC)N1C2=C(NC(=N2)C3CCCC3)C(=O)N(CCC)C1=O
Relative Density.	1.195g/cm3

Storage & Solubility Information

Storage

keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

Ethanol: < 1 mg/mL (insoluble or slightly soluble)

DMSO: 3.05 mg/mL (10.02 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.2853 mL	16.4263 mL	32.8526 mL	164.2630 mL
5 mM	0.6571 mL	3.2853 mL	6.5705 mL	32.8526 mL
10 mM	0.3285 mL	1.6426 mL	3.2853 mL	16.4263 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc