Shopping Cart
Remove All
  • TargetMol
    Your shopping cart is currently empty

DPCPX

🥰Excellent
Catalog No. T22744Cas No. 102146-07-6
Alias PD 116948

DPCPX (PD 116948) is an A1 adenosine receptor antagonist

DPCPX

DPCPX

🥰Excellent
Purity: 99.93%
Catalog No. T22744Alias PD 116948Cas No. 102146-07-6
DPCPX (PD 116948) is an A1 adenosine receptor antagonist
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
5 mg$31In StockIn Stock
10 mg$41In StockIn Stock
25 mg$65In StockIn Stock
50 mg$98In StockIn Stock
1 mL x 10 mM (in DMSO)$45In StockIn Stock
Add to Cart
Add to Quotation
In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
Questions
TargetMol
View More

Batch Information

Select Batch
Purity:99.93%
Appearance:Solid
Color:White
Contact us for more batch information

Resource Download

Product Introduction

Bioactivity
Description
DPCPX (PD 116948) is an A1 adenosine receptor antagonist
Targets&IC50
[3H]-CHA binding to A1 receptor (rat whole brain membranes):0.46 nM (Ki), [3H]-NECA binding to A2 receptor (rat striatal membranes):340 nM (Ki)
In vivo
DPCPX, a selective adenosine A1 receptor antagonist, enhances the antidepressant-like effects of imipramine, escitalopram, and reboxetine in mice behavioral tests
SynonymsPD 116948
Chemical Properties
Molecular Weight304.39
FormulaC16H24N4O2
Cas No.102146-07-6
SmilesC(CC)N1C2=C(NC(=N2)C3CCCC3)C(=O)N(CCC)C1=O
Relative Density.1.195g/cm3
Storage & Solubility Information
Storagekeep away from moisture | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
Ethanol: < 1 mg/mL (insoluble or slightly soluble)
DMSO: 3.05 mg/mL (10.02 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM3.2853 mL16.4263 mL32.8526 mL164.2630 mL
5 mM0.6571 mL3.2853 mL6.5705 mL32.8526 mL
10 mM0.3285 mL1.6426 mL3.2853 mL16.4263 mL

Calculator

  • Molarity Calculator
  • Dilution Calculator
  • Reconstitution Calculator
  • Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
TargetMol | Animal experiments For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent 10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.
Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSOTargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSOTargetMol | reagent stock solution to 400 μL PEG300TargetMol | reagent and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH2OTargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
% Tween 80
% Saline/PBS/ddH2O

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Related Tags: buy DPCPX | purchase DPCPX | DPCPX cost | order DPCPX | DPCPX chemical structure | DPCPX in vivo | DPCPX formula | DPCPX molecular weight