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VPC171

Name: VPC171
Brand: TargetMol
SKU: T29112
Price: 47 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T29112Cas No. 1018830-99-3

Alias VPC-171, VPC 171

VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).

VPC171

🥰Excellent

Purity: 99.78%

Catalog No. T29112Alias VPC-171, VPC 171Cas No. 1018830-99-3

VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).

Pack Size	Price	Availability
1 mg	$47	In Stock
5 mg	$93	In Stock
10 mg	$133	In Stock
25 mg	$247	In Stock
50 mg	$343	In Stock
100 mg	$487	In Stock
200 mg	$657	In Stock
1 mL x 10 mM (in DMSO)	$95	In Stock

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Batch Information

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Purity:99.78%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).
In vivo	VCP171 produced a greater inhibition of eEPSC amplitude of nerve-injury versus control animals in both lamina I and lamina II neurons[2].
Synonyms	VPC-171, VPC 171

Chemical Properties

Molecular Weight	347.35
Formula	C₁₈H₁₂F₃NOS
Cas No.	1018830-99-3
Smiles	Nc1scc(c1C(=O)c1ccccc1)-c1cccc(c1)C(F)(F)F
Relative Density.	1.345 g/cm3 (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 55 mg/mL (158.34 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.8789 mL	14.3947 mL	28.7894 mL	143.9470 mL
5 mM	0.5758 mL	2.8789 mL	5.7579 mL	28.7894 mL
10 mM	0.2879 mL	1.4395 mL	2.8789 mL	14.3947 mL
20 mM	0.1439 mL	0.7197 mL	1.4395 mL	7.1974 mL
50 mM	0.0576 mL	0.2879 mL	0.5758 mL	2.8789 mL
100 mM	0.0288 mL	0.1439 mL	0.2879 mL	1.4395 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc