keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Z-Gly-Pro-Phe-Leu-CHO (Z-GPFL-CHO) is a tetrapeptide aldehyde serving as a selective and potent proteasome inhibitor, demonstrating inhibition constants (Ki) of 1.5 µM, 2.3 µM, and 40.5 µM for branched-chain amino acid-preferred, small neutral amino acid-preferred, and chymotrypsin-like activities, respectively, and an inhibitory concentration (IC50) of 3.1 µM for peptidyl-glutamyl peptide hydrolyzing activity [1].
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Description | Z-Gly-Pro-Phe-Leu-CHO (Z-GPFL-CHO) is a tetrapeptide aldehyde serving as a selective and potent proteasome inhibitor, demonstrating inhibition constants (Ki) of 1.5 µM, 2.3 µM, and 40.5 µM for branched-chain amino acid-preferred, small neutral amino acid-preferred, and chymotrypsin-like activities, respectively, and an inhibitory concentration (IC50) of 3.1 µM for peptidyl-glutamyl peptide hydrolyzing activity [1]. |
Synonyms | Z-GPFL-CHO |
Molecular Weight | 550.65 |
Formula | C30H38N4O6 |
CAS No. | 159659-05-9 |
keep away from moisture
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Z-Gly-Pro-Phe-Leu-CHO 159659-05-9 Proteases/Proteasome Ubiquitination Proteasome Z-GPFL-CHO inhibitor inhibit