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Imidazoline Receptor

Imidazoline receptors are the primary receptors on which clonidine and other imidazolines act. There are three main classes of imidazoline receptors: I1 is involved in the inhibition of the sympathetic nervous system to lower blood pressure, I2 has as yet uncertain functions but is implicated in several psychiatric conditions, and I3 regulates insulin secretion.

  • Allantoin
    T092597-59-6
    Allantoin (Glyoxyldiureide), a urea hydantoin found in urine and plants, is used in dermatological preparations.
    • $50
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  • CR4056
    T150101004997-71-0
    CR4056 (6-(1H-imidazol-1-yl)-2-phenylquinazoline) is a selective inhibitor of MAO-A with IC50 of 202.7 nM and a ligand of I2-imidazoline receptor with IC50 of 596 nM.
    • $195
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    TargetMol | Inhibitor Sale
  • Harmane
    T3158486-84-0
    Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
    • $49
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    TargetMol | Citations Cited
  • BU 226 hydrochloride
    T220521186195-56-1
    BU 226 hydrochloride demonstrates affinity for imidazoline (I) receptors, in particular the I2 binding site with a Ki of 1.4 nM. BU 226 hydrochloride showed low (microM) affinity for alpha 2-adrenoceptors.
    • $53
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  • BU 224 hydrochloride
    T22051205437-64-5
    BU 224 hydrochloride is a selective imidazoline I(2) binding site ligand and has antinociceptive and antidepressant-like activities.
    • $34
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  • Rilmenidine hemifumarate
    T21911207572-68-7
    Rilmenidine hemifumarate (S-3341 hemifumarate) is a novel, orally active and selective I1 imidazoline receptor and α2-adrenoceptor agonist that induces autophagy, regulates the proliferation of leukaemia cells, stimulates the pro-apoptotic protein Bax, and induces autophagy in human leukaemia K5 cells. induces disruption of the mitochondrial pathway and apoptosis in human leukaemia K562 cells.
    • $72
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  • Rilmenidine Phosphate
    T664185409-38-7
    Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.
    • $34
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  • Agmatine sulfate
    T48082482-00-0
    Agmatine sulfate (Agmatine sulfate salt) is a bioactive metabolite of the arginine amino acid. It exerts modulatory action at multiple molecular targets, such as neurotransmitter systems, ion channels and nitric oxide synthesis. It is an endogenous agonist at imidazoline receptor and a NO synthase inhibitor.
    • $41
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  • Idazoxan hydrochloride
    T011579944-56-2
    Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
    • $43
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  • Moxonidine
    T102875438-57-2
    Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.
    • $33
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  • 2-BFI hydrochloride
    T2249289196-95-2
    2-BFI hydrochloride is a high-affinity agonist of I2-imidazoline receptor. 2-BFI hydrochloride can be used in studies about protection against stroke and acute inflammatory immune disease.
    • $53
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