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PKG inhibitor peptide TFA (82801-73-8 free base)

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Catalog No. TP1523
Alias PKG inhibitor peptide TFA

PKG inhibitor peptide TFA (82801-73-8 free base) is an inhibitor of ATP-competitive cGMP-dependent protein kinase (PKG).

PKG inhibitor peptide TFA (82801-73-8 free base)
Other Forms of PKG inhibitor peptide TFA (82801-73-8 free base):

PKG inhibitor peptide TFA (82801-73-8 free base)

🥰Excellent
Catalog No. TP1523Alias PKG inhibitor peptide TFA
PKG inhibitor peptide TFA (82801-73-8 free base) is an inhibitor of ATP-competitive cGMP-dependent protein kinase (PKG).
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$50In StockIn Stock
2 mg$70In StockIn Stock
5 mg$98In StockIn Stock
10 mg$141In StockIn Stock
25 mg$253In StockIn Stock
50 mg$381In StockIn Stock
100 mg$573In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction

Bioactivity
Description
PKG inhibitor peptide TFA (82801-73-8 free base) is an inhibitor of ATP-competitive cGMP-dependent protein kinase (PKG).
Targets&IC50
PKG: 86 μM(ki)
In vitro
PKG inhibitor peptide TFA binds to cGMP-dependent protein kinase directly with a Ki of 86 μM[1].
SynonymsPKG inhibitor peptide TFA
Chemical Properties
Molecular Weight1057.13
FormulaC40H75F3N18O12
SmilesC[C@@H](C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CCCN=C(N)N)N.C(=O)(C(F)(F)F)O
Relative Density.no data available
ColorWhite
Appearancesolid
Sequence{Arg}{Lys}{Arg}{Ala}{Arg}{Lys}{Glu}
Sequence ShortRKRARKE
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 10 mM, Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM0.9460 mL4.7298 mL9.4596 mL47.2979 mL
5 mM0.1892 mL0.9460 mL1.8919 mL9.4596 mL
10 mM0.0946 mL0.4730 mL0.9460 mL4.7298 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

PKG inhibitor peptide TFA (82801738 free base)PKG inhibitor peptide TFA (82801 73 8 free base)PKG82801-73-8 free base82801-73-8
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