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Pitavastatin lactone

🥰Excellent
Catalog No. T12490Cas No. 141750-63-2

Pitavastatin lactone is the major metabolite of Pitavastatin in humans.Pitavastatin is a competitive inhibitor of HMG-CoA reductase.

Pitavastatin lactone

Pitavastatin lactone

🥰Excellent
Purity: 98.18%
Catalog No. T12490Cas No. 141750-63-2
Pitavastatin lactone is the major metabolite of Pitavastatin in humans.Pitavastatin is a competitive inhibitor of HMG-CoA reductase.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
5 mg$39In StockIn Stock
10 mg$59In StockIn Stock
25 mg$128In StockIn Stock
50 mg$198In StockIn Stock
100 mg$297In StockIn Stock
200 mg$446In StockIn Stock
1 mL x 10 mM (in DMSO)$58In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Batch Information

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Purity:98.18%
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COA LCMS HNMR

Product Introduction

Bioactivity
Description
Pitavastatin lactone is the major metabolite of Pitavastatin in humans.Pitavastatin is a competitive inhibitor of HMG-CoA reductase.
Chemical Properties
Molecular Weight403.45
FormulaC25H22FNO3
Cas No.141750-63-2
SmilesC(=C/[C@@H]1C[C@@H](O)CC(=O)O1)\C2=C(C3=C(N=C2C4CC4)C=CC=C3)C5=CC=C(F)C=C5
Relative Density.1.372 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 60 mg/mL (148.72 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.4786 mL12.3931 mL24.7862 mL123.9311 mL
5 mM0.4957 mL2.4786 mL4.9572 mL24.7862 mL
10 mM0.2479 mL1.2393 mL2.4786 mL12.3931 mL
20 mM0.1239 mL0.6197 mL1.2393 mL6.1966 mL
50 mM0.0496 mL0.2479 mL0.4957 mL2.4786 mL
100 mM0.0248 mL0.1239 mL0.2479 mL1.2393 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
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Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Pitavastatin lactonepitavastatinmicrosomesmetaboliteInhibitorinhibithumansHMGCoAReductaseHMG-CoA reductaseHMGCoA ReductaseHMG-CoAhepaticDrug Metabolite
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