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TargetMol | Compound Library

Neurotransmitter Receptor Compound Library

Catalog No. L2610

A neurotransmitter receptor (also known as a neuroreceptor) is a membrane receptor protein that is activated by a neurotransmitter. Chemicals on the outside of the cell, such as a neurotransmitter, can bump into its corresponding receptor in the membrane, bind and trigger other events to occur inside the cell. A neurotransmitter receptor is a class of receptors that specifically binds with neurotransmitters as opposed to other molecules. Neurotransmitter (NT) receptors are located on the surface of neuronal and glial cells. There are two major types of neurotransmitter receptors: ionotropic and metabotropic. Ionotropic means that ions can pass through the receptor, whereas metabotropic means that a second messenger inside the cell relays the message (i.e. metabotropic receptors do not have channels). Metabotropic receptors are in fact G protein-coupled receptors. Ionotropic receptors are also called Ligand-gated ion channels and they can be excited by neurotransmitters like glutamate and aspartate. There are several major classes of neurotransmitters: Adrenergic, Dopaminergic, GABAergic, Glutaminergic, Histaminergic, Cholinergic, Opioid, Serotonergic, and Glycinergic. In the brain, most drug targets consist of signaling proteins that go awry in central nervous system diseases, for example with autism in childhood, schizophrenia in adolescence, or Alzheimer's disease in old age. The aim of drug treatment is to correct the inappropriate behavior of these proteins and restore normal brain function. Understanding the effects of neurotransmitters is extremely important in therapeutics. All psychiatric drugs act by affecting neurotransmitters. Understanding their mechanism of action and adverse effects is key to developing new drugs for neurological diseases. The TargetMol neurotransmitter receptor compound library contains 1513 CNS receptor ligands, which is ideal for screening or identifying recombinant orphan G protein-coupled receptors, target validation, secondary screening, validating new assays, and for routine pharmacological applications.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2610

Neurotransmitter Receptor Compound Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;
  • Targets include 5-HT receptor, AChR, GABA receptor, dopamine receptor,Opiod receptor, Ionotropic Glutamatergic receptor, Metabotropic Glutamatergic receptor, Purinergic receptor, etc.;
  • Structurally diverse, medicinally active, and cell permeable;
  • Detailed information about compound structure, target, activity, etc.;
  • NMR and HPLC/LCMS validated to ensure high purity and quality.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

5-HT Receptor
AChR
Dopamine Receptor
Adrenergic Receptor
Histamine Receptor
GABA Receptor
GluR
Adenosine Receptor
Opioid Receptor
AChE
iGluR
NMDAR
Autophagy
Endogenous Metabolite
Apoptosis
Norepinephrine
Serotonin Transporter
Antibacterial
Calcium Channel
Potassium Channel
Parasite
Sodium Channel
Neuropeptide Y Receptor
Endothelin Receptor
P450
PDE
Influenza Virus
NF-κB
HIV Protease
Antifungal
CaMK
cholecystokinin
Antibiotic
Reactive Oxygen Species
COX
HDAC
Phospholipase
HCV Protease
Mitophagy
TRP/TRPV Channel
P-gp
TNF
Histone Methyltransferase
Dehydrogenase
Ferroptosis
Virus Protease
ERK
MAO
Monoamine Transporter
DNA/RNA Synthesis
Beta Amyloid
Adenosine deaminase
Sigma receptor
NO Synthase
Chloride channel
Transferase
PI3K
BACE
RAAS
ABC
VEGFR
Caspase
Glucocorticoid Receptor
Drug Metabolite
P2X Receptor
HSV
Beta-Secretase
Prostaglandin Receptor
GPR
AMPK
Cannabinoid Receptor
Tyrosinase
Monoamine Oxidase
Adenylyl cyclase
NOS
Transaminase
Antioxidant
DYRK
Phosphatase
GSK-3
Melatonin Receptor
MRP
PKA
HBV
PPAR
PARP
PAFR
Gamma-secretase
ROS
BCL
IL Receptor
Aurora Kinase
cAMP
Lipoxygenase
mTOR
SARS-CoV
RSV
MEK
Anti-infection
Imidazoline Receptor
HER
Melanin-concentrating Hormone Receptor (MCHR)
CAT
Carbonic Anhydrase
Integrin
Amino Acids and Derivatives
p38 MAPK
Estrogen/progestogen Receptor
Na+/Ca2+ Exchanger
Arrestin
NADPH
GTPase
Progesterone Receptor
OCT
Antifolate
FXR
Leukotriene Receptor
PKC
Aryl Hydrocarbon Receptor
IAP
Immunology/Inflammation related
Annexin A
Adiponectin receptor
Bcr-Abl
LDL
GRK
Raf
MT Receptor
GlyT
Glucosidase
Mitochondrial Metabolism
Antifection
Fatty Acid Synthase
Bombesin Receptor
Stearoyl-CoA Desaturase (SCD)
CCR
MMP
PAD
ACK
Epigenetic Reader Domain
DNA
Indoleamine 2,3-Dioxygenase (IDO)
Androgen Receptor
Interleukin
TGF-beta/Smad
EGFR
Akt
MAPK
Acyltransferase
Trk receptor
Aminopeptidase
Nrf2
GluCls
GST
Reverse Transcriptase
STAT
CRISPR/Cas9
Hydroxylase
FGFR
Gap Junction Protein
Platelet aggregation
FLT
Syk
NOD
DNA Methyltransferase
HMG-CoA Reductase
Microtubule Associated
HIF/HIF Prolyl-Hydroxylase
FAK
p53

Keywords