Powder: -20°C for 3 years | In solvent: -80°C for 1 year
LSD1-IN-22 is a potent inhibitor of Lysine-specific demethylase 1 ( LSD1 ) with a K i value of 98 nM. LSD1-IN-22 has anti-proliferative activity against certain cancer cells [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 10-14 weeks | $ 1,520.00 | |
50 mg | 10-14 weeks | $ 1,980.00 | |
100 mg | 10-14 weeks | $ 2,500.00 |
Description | LSD1-IN-22 is a potent inhibitor of Lysine-specific demethylase 1 ( LSD1 ) with a K i value of 98 nM. LSD1-IN-22 has anti-proliferative activity against certain cancer cells [1]. |
In vitro | LSD1-IN-22 (compound 7t) demonstrates anti-proliferative effects on CCRF-CEM, Jurkat, and hERG cells. Utilizing a Cell Proliferation Assay across concentrations ranging from 0 to 50 μM over a period of 72 hours, results indicate significant inhibition of cell growth, with IC50 values of 23±0.8 μM for CCRF-CEM, 26±1.7 μM for Jurkat, and 7.7±1.3 μM for hERG cells. |
Molecular Weight | 248.07 |
Formula | C9H8BrF2N |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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