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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Citations

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
Antibiotic
COX
PI3K
Parasite
Adrenergic Receptor
EGFR
Ras
Calcium Channel
HIV Protease
AChR
Dopamine Receptor
VEGFR
PDE
Dehydrogenase
Cytochromes P450
ROS
Potassium Channel
Histamine Receptor
Epigenetic Reader Domain
Sodium Channel
Histone Methyltransferase
p38 MAPK
HDAC
ERK
Phosphatase
Antifungal
Akt
mTOR
JAK
Virus Protease
SARS-CoV
Src
FLT
Microtubule Associated
Cholinesterase (ChE)
Wnt/beta-catenin
STAT
iGluR
Influenza Virus
PARP
TNF
PDGFR
Reactive Oxygen Species
TRP/TRPV Channel
Topoisomerase
Prostaglandin Receptor
Caspase
FGFR
GSK-3
Raf
Interleukin
PKC
NO Synthase
Bcl-2 Family
HCV Protease
c-Kit
Monoamine Oxidase
MMP
c-Met/HGFR
GABA Receptor
Proteasome
RAAS
JNK
MAO
Lipoxygenase
Bcr-Abl
TGF-beta/Smad
Ferroptosis
ALK
HSP
MAPK
Phospholipase
E1/E2/E3 Enzyme
Transferase
Adenosine Receptor
NMDAR
DUB
GluR
Histone Demethylase
Drug Metabolite
PPAR
Tyrosinase
Beta Amyloid
Aurora Kinase
GPCR
Serine Protease
Integrin
ROCK
Kras
MDM-2/p53
HIF/HIF Prolyl-Hydroxylase
Casein Kinase
Reductase
PKA
Serotonin Transporter
AMPK
Anti-infection
Tyrosine Kinases
CCR
MEK
Mitochondrial Metabolism
IL Receptor
IκB/IKK
HSV
Serine/threonin kinase
ATPase
Reverse Transcriptase
Carbonic Anhydrase
Nucleoside Antimetabolite/Analog
P-gp
Mitophagy
Angiotensin-converting Enzyme (ACE)
HBV
Antiviral
Estrogen Receptor/ERR
Androgen Receptor
IGF-1R
Sirtuin
Cysteine Protease
TLR
CXCR
RIP kinase
Histone Acetyltransferase
Antioxidant
Proton pump
Glucosidase
Acyltransferase
c-RET
CaMK
DNA-PK
TAM Receptor
FAK
S6 Kinase
glycosidase
Leukotriene Receptor
NOD-like Receptor (NLR)
Gamma-secretase
NOS
Norepinephrine
LPL Receptor
P2X Receptor
HIF
Trk receptor
c-Fms
Estrogen/progestogen Receptor
PERK
Cannabinoid Receptor
ATM/ATR
FAAH
Nrf2
Hedgehog/Smoothened
NADPH
Immunology/Inflammation related
Chk
Glucocorticoid Receptor
Opioid Receptor
HER
Fatty Acid Synthase
Kinesin
PLK
Neurokinin receptor
p53
DPP-4
IDO
Indoleamine 2,3-Dioxygenase (IDO)
Syk
Pim
HMG-CoA Reductase
DYRK
NOD
Lipase
Endothelin Receptor
PD-1/PD-L1
transporter
PDK
Chloride channel
Glutathione Peroxidase
Antifection
DNA Methyltransferase
SGLT
Xanthine Oxidase
Smo
Hydroxylase
Aryl Hydrocarbon Receptor
Sigma receptor
Rho
IRAK
LTR
MAGL
LRRK2
ROS Kinase
YAP
Glutaminase
Thrombin
Mdm2
BTK
Isocitrate Dehydrogenase (IDH)
PAK
P2Y Receptor
IAP
Stearoyl-CoA Desaturase (SCD)
DHFR
PGE Synthase
Factor Xa
c-Myc
S1P Receptor
Retinoid Receptor
cAMP
Amino Acids and Derivatives
BACE
Epoxide Hydrolase
Cholecystokinin Receptor
Myosin
Beta-Secretase
MRP
Antifolate
OX Receptor
Aminopeptidase
PI4K
LPA Receptor
IRE1
Glucokinase
Complement System
Neuropeptide Y Receptor
Monocarboxylate transporter
OXPHOS
CSF-1R
Ephrin Receptor
RSV
ribosome
Telomerase
Lipid
AhR
GTPase
PAI-1
Aromatase
Monoamine Transporter
DNA
BCRP
Survivin
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Ligands for Target Protein for PROTAC
PAFR
ABC Transporter
Tie-2
CFTR
Adenylate cyclase
MLK
GST
Dynamin
ADC Cytotoxin
Necroptosis
GRK
STING
Acetyl-CoA Carboxylase
NADPH-oxidase
Vasopressin Receptor
Platelet aggregation
MicroRNA
Molecular Glues
DNA gyrase
Bradykinin Receptor
Pyroptosis
Neprilysin
MIF
OAT
MNK
ATP Citrate Lyase
Porcupine
SGK
MyD88
FLAP
CRM1
Neurotensin Receptor
PYK2
UGT
GlyT
Wee1
Methionine Adenosyltransferase (MAT)
p97
Na+/Ca2+ Exchanger
GNRH Receptor
NAMPT
Carboxypeptidase
Melanocortin Receptor
LIM Kinase
Glucagon Receptor
Phosphorylase
Prolyl Endopeptidase (PREP)
CGRP Receptor
SIK
IKZF
APC/C
PAD
ASK
DAPK
CRFR
Gap Junction Protein
MTP
PROTACs
cGAS
IFNAR
Bcl-6
Arp2/3 Complex
LDL
PTEN
GPX
LDLR
DNA Alkylation
Ligands for E3 Ligase
Protease
Hippo pathway
Arrestin
Melatonin Receptor
Guanylate cyclase
AAK1
Aquaporin
Progesterone Receptor
MELK
ROR
NEDD8
ATG
NR4A
CD73
CRISPR/Cas9
CETP
MT Receptor
Bombesin Receptor
MALT
DprE1
DNA Alkylator/Crosslinker
FXR
Amylase
Thyroid hormone receptor(THR)
Succinate Receptor 1 (SUCNR1)
Decarboxylase
FOXO
Adenosine Deaminase
BMI-1
CaSR
Liver X Receptor
HCN Channel
Oxytocin Receptor
Galectin
MTH1
KLF
CD38
VDAC
Vitamin
p62
Advanced Glycation End Products
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
ACK1
FKBP
Melanin-concentrating Hormone Receptor (MCHR)
NPC1L1
TOPK
Imidazoline Receptor
ASBT
PKM
Hexokinase
Orphan Receptor
Factor VIIa
Endonuclease
PROTAC Linker
TSH Receptor
Hck
HuR
FABP
KSP
Cadherin
Transaminase
Somatostatin
CAT
Arginase
ASCT
AIM2
GHSR
Apelin receptor
Haspin Kinase
GPCR19
PGK1
Ferroportin
Transketolase
NUDIX hydrolase
RANKL/RANK
Annexin A
PSMA
hCE
Huntingtin
Kisspeptin
Neuropeptide FF Receptor
Integrase
Glutaminyl Cyclase
Urea Transporter
GSNOR
EBI2/GPR183
Y Box Binding Protein 1
gp120/CD4
PARG（Poly(ADP-ribose) Glycohydrolase）
FOXO3
Drug-Linker Conjugates for ADC
stilbene oxidase
VDA
N-Acetylglucosaminyltransferase
Target Protein Ligand-Linker Conjugates
LAG-3
Photosystem (PS)
Adiponectin Receptor
Anion Exchanger
E3 Ligase Ligand-Linker Conjugates
CD74
Piezo Channel
Procollagen C Proteinase
Cell wall
OCT
Stemness kinase
Fas/FasL
Early 2 Factor (E2F)
RAR/RXR
Neuropeptide W
PACAP
MRGPR
GluCls
Glyoxalase
Taste receptor
Aconitase
Thioredoxin
Glutathione reductase
Mucin
Cuproptosis
LHRH
Photosensitizer
CPT
REV-ERB
Lysosomal Autophagy
NEDD4-1
Fer/FerT kinase
Tight Junction Protein
Poly(ADP-ribose) Glycohydrolase (PARG)
Sodium-dependent phosphate transporter
PGC-1α
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