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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

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Targetmol Compound Libraries
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
Endogenous Metabolite
CDK
DNA/RNA Synthesis
Antibiotic
COX
NF-κB
AChR
EGFR
PI3K
Ras
Parasite
HIV Protease
Adrenergic Receptor
Dopamine Receptor
Calcium Channel
PDE
VEGFR
Dehydrogenase
Epigenetic Reader Domain
Potassium Channel
Histamine Receptor
Cytochromes P450
Sodium Channel
Histone Methyltransferase
HDAC
Antifungal
Phosphatase
JAK
mTOR
Virus Protease
Src
p38 MAPK
SARS-CoV
Akt
FLT
ERK
Microtubule Associated
PARP
Cholinesterase (ChE)
Reactive Oxygen Species
TRP/TRPV Channel
Topoisomerase
PDGFR
Influenza Virus
iGluR
PKC
STAT
FGFR
Wnt/beta-catenin
Raf
Prostaglandin Receptor
TNF
HCV Protease
GSK-3
Bcl-2 Family
c-Kit
c-Met/HGFR
GABA Receptor
Monoamine Oxidase
Proteasome
Caspase
MAO
RAAS
MMP
Bcr-Abl
Lipoxygenase
NO Synthase
ALK
Ferroptosis
TGF-beta/Smad
HSP
NMDAR
Adenosine Receptor
MAPK
Phospholipase
DUB
Transferase
GluR
Interleukin
Histone Demethylase
Aurora Kinase
GPCR
JNK
E1/E2/E3 Enzyme
Beta Amyloid
Tyrosinase
Kras
PPAR
ROCK
Anti-infection
Tyrosine Kinases
Serine Protease
Drug Metabolite
HIF/HIF Prolyl-Hydroxylase
Integrin
Casein Kinase
Serotonin Transporter
AMPK
ATPase
IL Receptor
PKA
Mitochondrial Metabolism
CCR
IκB/IKK
MEK
Reductase
Serine/threonin kinase
Reverse Transcriptase
Carbonic Anhydrase
HSV
MDM-2/p53
Mitophagy
Antiviral
Nucleoside Antimetabolite/Analog
Cysteine Protease
Angiotensin-converting Enzyme (ACE)
Androgen Receptor
HBV
Glucosidase
Sirtuin
Estrogen Receptor/ERR
IGF-1R
Histone Acetyltransferase
Antioxidant
c-RET
DNA-PK
RIP kinase
ROS
Proton pump
CXCR
S6 Kinase
TAM Receptor
Acyltransferase
TLR
Norepinephrine
P-gp
HIF
Estrogen/progestogen Receptor
LPL Receptor
Leukotriene Receptor
Gamma-secretase
P2X Receptor
CaMK
c-Fms
FAK
NOS
FAAH
Opioid Receptor
Trk receptor
ATM/ATR
NADPH
DPP-4
PLK
Cannabinoid Receptor
NOD-like Receptor (NLR)
HER
Immunology/Inflammation related
Hedgehog/Smoothened
Neurokinin receptor
Syk
p53
Glucocorticoid Receptor
Chk
Pim
Fatty Acid Synthase
NOD
HMG-CoA Reductase
DYRK
Endothelin Receptor
DNA Methyltransferase
Chloride channel
PERK
IDO
Antifection
Indoleamine 2,3-Dioxygenase (IDO)
Kinesin
Smo
transporter
Nrf2
Glutathione Peroxidase
SGLT
Hydroxylase
IRAK
PD-1/PD-L1
LTR
Rho
MAGL
LRRK2
PDK
Sigma receptor
ROS Kinase
P2Y Receptor
Lipase
Aryl Hydrocarbon Receptor
BTK
PAK
Xanthine Oxidase
DHFR
Factor Xa
Isocitrate Dehydrogenase (IDH)
PGE Synthase
Thrombin
S1P Receptor
Mdm2
YAP
BACE
c-Myc
Glutaminase
IAP
Myosin
cAMP
Retinoid Receptor
MRP
Cholecystokinin Receptor
OX Receptor
Epoxide Hydrolase
Amino Acids and Derivatives
Glucokinase
IRE1
Stearoyl-CoA Desaturase (SCD)
Beta-Secretase
Aminopeptidase
LPA Receptor
PI4K
Complement System
Antifolate
CSF-1R
Ephrin Receptor
ribosome
GTPase
Monoamine Transporter
Neuropeptide Y Receptor
Telomerase
RSV
Aromatase
AhR
Monocarboxylate transporter
Ligands for Target Protein for PROTAC
DNA
OXPHOS
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Tie-2
ABC Transporter
Lipid
PAI-1
GST
ADC Cytotoxin
MicroRNA
PAFR
Vasopressin Receptor
BCRP
Acetyl-CoA Carboxylase
Platelet aggregation
NADPH-oxidase
CFTR
MLK
Dynamin
MIF
GRK
DNA gyrase
Bradykinin Receptor
MNK
Survivin
Neprilysin
Melanocortin Receptor
CRM1
Na+/Ca2+ Exchanger
GNRH Receptor
Neurotensin Receptor
LIM Kinase
NAMPT
PYK2
FLAP
Molecular Glues
Wee1
OAT
Porcupine
STING
Methionine Adenosyltransferase (MAT)
SGK
MyD88
Necroptosis
SIK
UGT
LDL
Glucagon Receptor
Phosphorylase
GlyT
PAD
ATP Citrate Lyase
ASK
CRFR
Pyroptosis
Carboxypeptidase
APC/C
p97
Adenylyl Cyclase
Bcl-6
AAK1
Prolyl Endopeptidase (PREP)
DNA Alkylation
PTEN
cGAS
GPX
Ligand for E3 Ligase
CGRP Receptor
DAPK
IKZF
ROR
MTP
IFNAR
Progesterone Receptor
Melatonin Receptor
Arp2/3 Complex
Guanylate cyclase
MELK
Hippo pathway
Protease
Aquaporin
Gap Junction Protein
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
PROTACs
MALT
NEDD8
DprE1
Succinate Receptor 1 (SUCNR1)
DNA Alkylator/Crosslinker
CETP
Galectin
CaSR
ATG
FXR
NR4A
Amylase
MTH1
MT Receptor
AAK1 (AP2 associated kinase 1)
Bombesin Receptor
CD73
Decarboxylase
KLF
CRISPR/Cas9
Oxytocin Receptor
Adenosine Deaminase
BMI-1
Advanced Glycation End Products
NPC1L1
CD38
ASBT
Arrestin
VDAC
LDLR
Hexokinase
HCN Channel
ACK1
p62
FKBP
Imidazoline Receptor
Apelin receptor
CAT
Transaminase
Arginase
Factor VIIa
TOPK
ASCT
Hck
Liver X Receptor
Endonuclease
Haspin Kinase
Na-K-Cl cotransporter
Somatostatin
Cadherin
GPCR19
AIM2
TSH Receptor
HuR
GHSR
FOXO
PKM
PGK1
GSNOR
NUDIX hydrolase
EBI2/GPR183
Y Box Binding Protein 1
Glutaminyl Cyclase
gp120/CD4
Kisspeptin
RANKL/RANK
Annexin A
Neuropeptide FF Receptor
FABP
Integrase
KSP
Transketolase
hCE
Vitamin
PARG（Poly(ADP-ribose) Glycohydrolase）
Drug-Linker Conjugates for ADC
FOXO3
Taste receptor
stilbene oxidase
RAR/RXR
Piezo Channel
Procollagen C Proteinase
Neuropeptide W
Aconitase
Cell wall
LHRH
VDA
OCT
N-Acetylglucosaminyltransferase
Photosensitizer
Stemness kinase
Photosystem (PS)
Adiponectin Receptor
Fas/FasL
PACAP
Anion Exchanger
PROTAC Linker
Thioredoxin
glycosidase
Mucin
Target Protein Ligand-Linker Conjugate
Huntingtin
PSMA
Glutathione reductase
MRGPR
Early 2 Factor (E2F)
Urea Transporter
CD74
CPT
GluCls
NEDD4-1
Cuproptosis
REV-ERB
Fer/FerT kinase
Tight Junction Protein
Lysosomal Autophagy
Glyoxalase
Ferroportin
Sodium-dependent phosphate transporter
Poly(ADP-ribose) Glycohydrolase (PARG)
PGC-1α
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