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TOPProduct DescriptionPackaging & StorageSupporting FilesLibrary CustomizationLibrary Composition
TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
Antibiotic
COX
PI3K
AChR
Parasite
Adrenergic Receptor
EGFR
Ras
Calcium Channel
HIV Protease
Dopamine Receptor
VEGFR
PDE
Potassium Channel
Dehydrogenase
ROS
Cytochromes P450
Histamine Receptor
Epigenetic Reader Domain
Sodium Channel
Histone Methyltransferase
p38 MAPK
HDAC
Antifungal
ERK
Phosphatase
Akt
mTOR
Virus Protease
JAK
SARS-CoV
Src
FLT
Microtubule Associated
Cholinesterase (ChE)
Influenza Virus
TNF
Wnt/beta-catenin
STAT
PARP
iGluR
PDGFR
Reactive Oxygen Species
TRP/TRPV Channel
Topoisomerase
Prostaglandin Receptor
FGFR
GSK-3
Caspase
Bcl-2 Family
PKC
Interleukin
NO Synthase
Raf
HCV Protease
c-Kit
Monoamine Oxidase
GABA Receptor
MMP
c-Met/HGFR
Proteasome
RAAS
MAO
JNK
Ferroptosis
Lipoxygenase
Bcr-Abl
TGF-beta/Smad
ALK
HSP
MAPK
Phospholipase
Adenosine Receptor
NMDAR
Transferase
DUB
E1/E2/E3 Enzyme
GluR
Histone Demethylase
PPAR
Drug Metabolite
Tyrosinase
Beta Amyloid
Aurora Kinase
GPCR
Serine Protease
Integrin
ROCK
Kras
Reductase
Serotonin Transporter
HIF/HIF Prolyl-Hydroxylase
Tyrosine Kinases
Casein Kinase
PKA
AMPK
Anti-infection
MDM-2/p53
CCR
Mitochondrial Metabolism
MEK
Serine/threonin kinase
ATPase
IκB/IKK
HSV
IL Receptor
Reverse Transcriptase
Carbonic Anhydrase
P-gp
Nucleoside Antimetabolite/Analog
Angiotensin-converting Enzyme (ACE)
HBV
IGF-1R
Mitophagy
Estrogen Receptor/ERR
Androgen Receptor
Antiviral
Cysteine Protease
Sirtuin
CXCR
TLR
Glucosidase
Histone Acetyltransferase
RIP kinase
Proton pump
Antioxidant
c-RET
glycosidase
Acyltransferase
TAM Receptor
CaMK
DNA-PK
FAK
S6 Kinase
Leukotriene Receptor
Norepinephrine
NOD-like Receptor (NLR)
HIF
PERK
Trk receptor
c-Fms
P2X Receptor
NOS
Gamma-secretase
Estrogen/progestogen Receptor
LPL Receptor
Cannabinoid Receptor
ATM/ATR
Nrf2
FAAH
Opioid Receptor
Hedgehog/Smoothened
Chk
NADPH
HER
Immunology/Inflammation related
DPP-4
PLK
Fatty Acid Synthase
Kinesin
Neurokinin receptor
Syk
p53
Indoleamine 2,3-Dioxygenase (IDO)
Pim
IDO
Glucocorticoid Receptor
DYRK
NOD
Lipase
Endothelin Receptor
PD-1/PD-L1
HMG-CoA Reductase
Chloride channel
Glutathione Peroxidase
Antifection
transporter
PDK
DNA Methyltransferase
Xanthine Oxidase
Smo
SGLT
IRAK
Aryl Hydrocarbon Receptor
Hydroxylase
Rho
MAGL
LRRK2
LTR
Sigma receptor
ROS Kinase
Thrombin
c-Myc
BTK
Isocitrate Dehydrogenase (IDH)
PAK
P2Y Receptor
YAP
Factor Xa
DHFR
S1P Receptor
Glutaminase
PGE Synthase
Stearoyl-CoA Desaturase (SCD)
Mdm2
cAMP
Retinoid Receptor
IAP
Myosin
Amino Acids and Derivatives
Epoxide Hydrolase
Cholecystokinin Receptor
Beta-Secretase
PI4K
MRP
Antifolate
OX Receptor
Aminopeptidase
BACE
IRE1
Glucokinase
Complement System
LPA Receptor
Ephrin Receptor
Monocarboxylate transporter
OXPHOS
Monoamine Transporter
CSF-1R
RSV
Neuropeptide Y Receptor
GTPase
PAI-1
Aromatase
ribosome
Telomerase
Lipid
AhR
DNA
Ligands for Target Protein for PROTAC
BCRP
Survivin
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
GST
Acetyl-CoA Carboxylase
MLK
ABC Transporter
CFTR
Tie-2
Dynamin
PAFR
ADC Cytotoxin
Vasopressin Receptor
Platelet aggregation
STING
NADPH-oxidase
MicroRNA
Necroptosis
GRK
Melanocortin Receptor
DNA gyrase
Bradykinin Receptor
Pyroptosis
Neprilysin
OAT
MNK
MIF
Molecular Glues
Na+/Ca2+ Exchanger
GNRH Receptor
NAMPT
Carboxypeptidase
MyD88
Porcupine
FLAP
LIM Kinase
Glucagon Receptor
CRM1
Neurotensin Receptor
PYK2
UGT
GlyT
Wee1
Methionine Adenosyltransferase (MAT)
p97
SGK
CRFR
Gap Junction Protein
Prolyl Endopeptidase (PREP)
LDL
CGRP Receptor
ATP Citrate Lyase
SIK
IKZF
APC/C
PAD
ASK
DAPK
Phosphorylase
MTP
PTEN
GPX
PROTACs
cGAS
LDLR
DNA Alkylation
Ligand for E3 Ligase
Protease
Adenylyl Cyclase
IFNAR
Bcl-6
Arp2/3 Complex
Progesterone Receptor
MELK
DNA Alkylator/Crosslinker
Arrestin
Melatonin Receptor
Guanylate cyclase
Hippo pathway
AAK1
ROR
Aquaporin
CaSR
Liver X Receptor
HCN Channel
Oxytocin Receptor
MALT
DprE1
FXR
Amylase
NEDD8
ATG
NR4A
CD73
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
Succinate Receptor 1 (SUCNR1)
Decarboxylase
FOXO
Adenosine Deaminase
Galectin
MTH1
KLF
CETP
MT Receptor
Bombesin Receptor
BMI-1
FKBP
CD38
VDAC
Vitamin
p62
CRISPR/Cas9
NPC1L1
TOPK
PKM
Imidazoline Receptor
Hexokinase
ASBT
Advanced Glycation End Products
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
ACK1
CAT
Arginase
ASCT
AIM2
GHSR
FABP
KSP
Cadherin
Factor VIIa
Endonuclease
TSH Receptor
Apelin receptor
Haspin Kinase
Orphan Receptor
GPCR19
Transaminase
Somatostatin
Hck
HuR
Ferroportin
PGK1
GSNOR
EBI2/GPR183
Y Box Binding Protein 1
gp120/CD4
Photosensitizer
Huntingtin
Transketolase
Kisspeptin
Neuropeptide FF Receptor
Integrase
Glutaminyl Cyclase
Urea Transporter
NUDIX hydrolase
RANKL/RANK
Annexin A
PSMA
hCE
PARG（Poly(ADP-ribose) Glycohydrolase）
Drug-Linker Conjugates for ADC
FOXO3
LHRH
CPT
REV-ERB
RAR/RXR
Neuropeptide W
PACAP
MRGPR
GluCls
stilbene oxidase
VDA
N-Acetylglucosaminyltransferase
LAG-3
Photosystem (PS)
Adiponectin Receptor
Anion Exchanger
PROTAC Linker
CD74
Taste receptor
Aconitase
Thioredoxin
Glutathione reductase
Lysosomal Autophagy
Glyoxalase
Target Protein Ligand-Linker Conjugate
NEDD4-1
Fer/FerT kinase
Tight Junction Protein
Mucin
Cuproptosis
Piezo Channel
Procollagen C Proteinase
Cell wall
OCT
Stemness kinase
Fas/FasL
Early 2 Factor (E2F)
Sodium-dependent phosphate transporter
Poly(ADP-ribose) Glycohydrolase (PARG)
PGC-1α
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