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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively. Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

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Targetmol Compound Libraries
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
CDK
COX
EGFR
AChR
Antibiotic
PI3K
DNA/RNA Synthesis
HIV Protease
Endogenous Metabolite
Adrenergic Receptor
Dopamine Receptor
PDE
NF-κB
Calcium Channel
VEGFR
Epigenetic Reader Domain
Dehydrogenase
Histamine Receptor
Potassium Channel
Histone Methyltransferase
Cytochromes P450
Sodium Channel
HDAC
Parasite
Phosphatase
Antifungal
JAK
mTOR
Src
FLT
Microtubule Associated
Topoisomerase
TRP/TRPV Channel
PDGFR
Cholinesterase (ChE)
SARS-CoV
PKC
FGFR
PARP
Wnt/beta-catenin
p38 MAPK
Raf
Akt
Influenza Virus
HCV Protease
ERK
STAT
c-Kit
GSK-3
MAO
Prostaglandin Receptor
RAAS
GABA Receptor
c-Met/HGFR
Lipoxygenase
Bcr-Abl
ALK
TNF
NMDAR
MMP
Proteasome
Adenosine Receptor
Reactive Oxygen Species
GluR
Bcl-2 Family
Ferroptosis
DUB
HSP
Phospholipase
Virus Protease
Histone Demethylase
Aurora Kinase
TGF-beta/Smad
Tyrosinase
Tyrosine Kinases
Ras
GPCR
MAPK
ROCK
IL Receptor
iGluR
Casein Kinase
ATPase
Transferase
Integrin
CCR
E1/E2/E3 Enzyme
Beta Amyloid
MEK
Monoamine Oxidase
Carbonic Anhydrase
JNK
PKA
PPAR
Antiviral
Serine/threonin kinase
Caspase
NO Synthase
Androgen Receptor
Reverse Transcriptase
Serotonin Transporter
IκB/IKK
Antioxidant
Mitophagy
Cysteine Protease
AMPK
Mitochondrial Metabolism
HSV
Sirtuin
DNA-PK
HBV
RIP kinase
c-RET
CXCR
TAM Receptor
Reductase
IGF-1R
Norepinephrine
HIF
NOS
P2X Receptor
ROS
Estrogen/progestogen Receptor
Estrogen Receptor/ERR
Nucleoside Antimetabolite/Analog
CaMK
P-gp
TLR
Histone Acetyltransferase
Serine Protease
Gamma-secretase
Drug Metabolite
Glucosidase
HIF/HIF Prolyl-Hydroxylase
Interleukin
DPP-4
FAAH
Trk receptor
c-Fms
S6 Kinase
FAK
HER
Proton pump
Hedgehog/Smoothened
Acyltransferase
ATM/ATR
PLK
p53
Opioid Receptor
Cannabinoid Receptor
Neurokinin receptor
Syk
Glucocorticoid Receptor
Fatty Acid Synthase
Endothelin Receptor
Chk
NOD
HMG-CoA Reductase
Pim
Immunology/Inflammation related
Kinesin
Chloride channel
DYRK
NADPH
Rho
SGLT
LTR
Leukotriene Receptor
Antifection
Indoleamine 2,3-Dioxygenase (IDO)
LRRK2
transporter
Anti-infection
DNA Methyltransferase
IRAK
LPL Receptor
PDK
Lipase
Factor Xa
Nrf2
Thrombin
PD-1/PD-L1
S1P Receptor
Kras
BTK
Mdm2
P2Y Receptor
BACE
PERK
Glutathione Peroxidase
Smo
Xanthine Oxidase
cAMP
Hydroxylase
Sigma receptor
DHFR
MRP
PAK
Epoxide Hydrolase
Retinoid Receptor
Cholecystokinin Receptor
Glucokinase
IRE1
OX Receptor
LPA Receptor
ROS Kinase
YAP
c-Myc
CSF-1R
ribosome
PI4K
Complement System
GTPase
Glutaminase
Aryl Hydrocarbon Receptor
IAP
Myosin
Ephrin Receptor
Aromatase
AhR
Antifolate
DNA
PGE Synthase
Aminopeptidase
Protease-activated Receptor
ABC Transporter
Monoamine Transporter
Isocitrate Dehydrogenase (IDH)
Neuropeptide Y Receptor
Telomerase
RSV
Discoidin Domain Receptor (DDR)
ADC Cytotoxin
MicroRNA
Monocarboxylate transporter
IDO
Stearoyl-CoA Desaturase (SCD)
Vasopressin Receptor
Beta-Secretase
Platelet aggregation
NADPH-oxidase
NOD-like Receptor (NLR)
GRK
DNA gyrase
Bradykinin Receptor
PAI-1
Neprilysin
Acetyl-CoA Carboxylase
Melanocortin Receptor
CFTR
MLK
Dynamin
GNRH Receptor
LIM Kinase
NAMPT
ATP Citrate Lyase
Lipid
BCRP
MNK
STING
Ligands for Target Protein for PROTAC
Neurotensin Receptor
SIK
LDL
Glucagon Receptor
Phosphorylase
GlyT
PAD
Wee1
OAT
Porcupine
ASK
GST
Carboxypeptidase
SGK
APC/C
Adenylyl Cyclase
Na+/Ca2+ Exchanger
Tie-2
MIF
Bcl-6
AAK1
PYK2
UGT
MAGL
DNA Alkylation
Angiotensin-converting Enzyme (ACE)
CRFR
GPX
p97
IKZF
ROR
MTP
CRM1
Amino Acids and Derivatives
Progesterone Receptor
FLAP
PAFR
MT Receptor
Guanylate cyclase
cGAS
MELK
Methionine Adenosyltransferase (MAT)
Ligand for E3 Ligase
Protease
CGRP Receptor
Gap Junction Protein
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
PROTACs
MALT
MyD88
DprE1
Succinate Receptor 1 (SUCNR1)
DNA Alkylator/Crosslinker
CETP
Amylase
MTH1
Bombesin Receptor
OXPHOS
Survivin
CD73
Decarboxylase
Hippo pathway
CRISPR/Cas9
Aquaporin
Adenosine Deaminase
DAPK
BMI-1
Advanced Glycation End Products
NPC1L1
CD38
NEDD8
Melatonin Receptor
Galectin
CaSR
VDAC
ATG
LDLR
Hexokinase
HCN Channel
ACK1
PTEN
Pyroptosis
Imidazoline Receptor
CAT
Transaminase
Arginase
Factor VIIa
Arrestin
IFNAR
Necroptosis
TOPK
ASCT
Hck
Liver X Receptor
NR4A
Haspin Kinase
KSP
Cadherin
TSH Receptor
HuR
Oxytocin Receptor
GHSR
PKM
PGK1
Apelin receptor
GSNOR
NUDIX hydrolase
EBI2/GPR183
Glutaminyl Cyclase
gp120/CD4
Kisspeptin
FXR
Prolyl Endopeptidase (PREP)
Neuropeptide FF Receptor
FABP
Na-K-Cl cotransporter
Molecular Glues
Integrase
Somatostatin
Transketolase
AIM2
hCE
p62
KLF
FOXO
Drug-Linker Conjugates for ADC
FOXO3
Taste receptor
stilbene oxidase
RAR/RXR
ASBT
Piezo Channel
Y Box Binding Protein 1
Procollagen C Proteinase
Aconitase
Neuropeptide W
Cell wall
LHRH
VDA
OCT
N-Acetylglucosaminyltransferase
Photosensitizer
Stemness kinase
RANKL/RANK
Adiponectin Receptor
Endonuclease
Fas/FasL
PACAP
Anion Exchanger
Thioredoxin
Mucin
Huntingtin
PSMA
Glutathione reductase
MRGPR
GPCR19
Urea Transporter
CD74
CPT
GluCls
NEDD4-1
Fer/FerT kinase
Tight Junction Protein
Lysosomal Autophagy
Glyoxalase
Sodium-dependent phosphate transporter
Vitamin
PARG（Poly(ADP-ribose) Glycohydrolase）
PGC-1α
Poly(ADP-ribose) Glycohydrolase (PARG)
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