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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
Antibiotic
COX
PI3K
Parasite
Adrenergic Receptor
EGFR
Ras
Calcium Channel
HIV Protease
AChR
Dopamine Receptor
VEGFR
PDE
Dehydrogenase
ROS
Cytochromes P450
Potassium Channel
Histamine Receptor
Epigenetic Reader Domain
Sodium Channel
Histone Methyltransferase
p38 MAPK
ERK
Phosphatase
HDAC
Antifungal
Akt
mTOR
JAK
Virus Protease
SARS-CoV
Src
FLT
Microtubule Associated
Cholinesterase (ChE)
Wnt/beta-catenin
STAT
iGluR
Influenza Virus
PARP
TNF
Reactive Oxygen Species
PDGFR
TRP/TRPV Channel
Topoisomerase
Caspase
Prostaglandin Receptor
GSK-3
FGFR
Raf
Interleukin
PKC
NO Synthase
Bcl-2 Family
HCV Protease
c-Kit
Monoamine Oxidase
MMP
c-Met/HGFR
GABA Receptor
Proteasome
RAAS
JNK
MAO
Lipoxygenase
Bcr-Abl
ALK
Ferroptosis
TGF-beta/Smad
HSP
MAPK
Phospholipase
Transferase
Adenosine Receptor
E1/E2/E3 Enzyme
NMDAR
DUB
PPAR
GluR
Histone Demethylase
Drug Metabolite
Tyrosinase
Aurora Kinase
Beta Amyloid
GPCR
Serine Protease
Integrin
ROCK
Kras
MDM-2/p53
HIF/HIF Prolyl-Hydroxylase
Reductase
PKA
Serotonin Transporter
Casein Kinase
AMPK
Anti-infection
Tyrosine Kinases
CCR
Mitochondrial Metabolism
MEK
IL Receptor
Serine/threonin kinase
IκB/IKK
HSV
ATPase
Carbonic Anhydrase
Reverse Transcriptase
Mitophagy
Nucleoside Antimetabolite/Analog
Angiotensin-converting Enzyme (ACE)
P-gp
Estrogen Receptor/ERR
HBV
Androgen Receptor
IGF-1R
Antiviral
Sirtuin
Cysteine Protease
TLR
RIP kinase
CXCR
Histone Acetyltransferase
Antioxidant
Glucosidase
Acyltransferase
c-RET
Proton pump
DNA-PK
CaMK
TAM Receptor
FAK
Leukotriene Receptor
Gamma-secretase
glycosidase
S6 Kinase
NOD-like Receptor (NLR)
NOS
LPL Receptor
P2X Receptor
Norepinephrine
Trk receptor
c-Fms
HIF
Estrogen/progestogen Receptor
PERK
ATM/ATR
Hedgehog/Smoothened
FAAH
Nrf2
Cannabinoid Receptor
NADPH
Chk
Glucocorticoid Receptor
Immunology/Inflammation related
Opioid Receptor
PLK
HER
Kinesin
DPP-4
Fatty Acid Synthase
Neurokinin receptor
p53
Pim
IDO
Indoleamine 2,3-Dioxygenase (IDO)
Syk
DYRK
Lipase
NOD
HMG-CoA Reductase
Endothelin Receptor
PD-1/PD-L1
Chloride channel
Glutathione Peroxidase
Antifection
transporter
PDK
DNA Methyltransferase
Smo
Xanthine Oxidase
SGLT
Rho
Aryl Hydrocarbon Receptor
Hydroxylase
IRAK
Sigma receptor
LTR
MAGL
LRRK2
Thrombin
ROS Kinase
Mdm2
YAP
P2Y Receptor
Glutaminase
BTK
Isocitrate Dehydrogenase (IDH)
PAK
S1P Receptor
DHFR
Factor Xa
c-Myc
IAP
Stearoyl-CoA Desaturase (SCD)
PGE Synthase
Amino Acids and Derivatives
cAMP
Retinoid Receptor
BACE
MRP
Cholecystokinin Receptor
Antifolate
Myosin
OX Receptor
Epoxide Hydrolase
Beta-Secretase
Aminopeptidase
Glucokinase
IRE1
LPA Receptor
PI4K
Complement System
Monocarboxylate transporter
CSF-1R
Neuropeptide Y Receptor
OXPHOS
Ephrin Receptor
RSV
GTPase
Telomerase
PAI-1
Aromatase
ribosome
AhR
Ligands for Target Protein for PROTAC
PAFR
Monoamine Transporter
DNA
Lipid
BCRP
Survivin
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Dynamin
Tie-2
Adenylate cyclase
ABC Transporter
GST
CFTR
MLK
ADC Cytotoxin
MicroRNA
Necroptosis
GRK
Vasopressin Receptor
STING
Acetyl-CoA Carboxylase
Platelet aggregation
NADPH-oxidase
MIF
DNA gyrase
Molecular Glues
Bradykinin Receptor
MNK
OAT
Pyroptosis
Neprilysin
CRM1
MyD88
Na+/Ca2+ Exchanger
GNRH Receptor
Neurotensin Receptor
NAMPT
PYK2
FLAP
UGT
Glucagon Receptor
GlyT
ATP Citrate Lyase
Wee1
Porcupine
Methionine Adenosyltransferase (MAT)
Carboxypeptidase
Melanocortin Receptor
SGK
p97
LIM Kinase
SIK
Phosphorylase
IKZF
PAD
ASK
CRFR
CGRP Receptor
Gap Junction Protein
DAPK
APC/C
MTP
PROTACs
IFNAR
Bcl-6
LDLR
Prolyl Endopeptidase (PREP)
LDL
Arp2/3 Complex
Ligands for E3 Ligase
DNA Alkylation
PTEN
cGAS
GPX
Protease
ROR
Arrestin
Progesterone Receptor
Melatonin Receptor
Guanylate cyclase
MELK
Hippo pathway
Aquaporin
Thyroid hormone receptor(THR)
MALT
NEDD8
DprE1
Succinate Receptor 1 (SUCNR1)
DNA Alkylator/Crosslinker
CETP
Galectin
CaSR
AAK1
ATG
Liver X Receptor
FXR
NR4A
Amylase
MTH1
MT Receptor
HCN Channel
Bombesin Receptor
CD73
Decarboxylase
KLF
CRISPR/Cas9
Oxytocin Receptor
FOXO
Adenosine Deaminase
BMI-1
Melanin-concentrating Hormone Receptor (MCHR)
Advanced Glycation End Products
NPC1L1
CD38
ASBT
TOPK
VDAC
Vitamin
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
Hexokinase
ACK1
Orphan Receptor
p62
FKBP
Imidazoline Receptor
PKM
Apelin receptor
CAT
Transaminase
Arginase
Factor VIIa
ASCT
Hck
Endonuclease
FABP
Haspin Kinase
PROTAC Linker
Somatostatin
KSP
Cadherin
GPCR19
AIM2
TSH Receptor
HuR
GHSR
Ferroportin
PGK1
GSNOR
NUDIX hydrolase
EBI2/GPR183
Y Box Binding Protein 1
Glutaminyl Cyclase
gp120/CD4
Kisspeptin
RANKL/RANK
Annexin A
Neuropeptide FF Receptor
Integrase
Transketolase
Huntingtin
PSMA
Urea Transporter
hCE
PARG（Poly(ADP-ribose) Glycohydrolase）
Drug-Linker Conjugates for ADC
FOXO3
Taste receptor
stilbene oxidase
RAR/RXR
Piezo Channel
Procollagen C Proteinase
Neuropeptide W
Aconitase
Cell wall
LHRH
VDA
OCT
N-Acetylglucosaminyltransferase
Photosensitizer
Target Protein Ligand-Linker Conjugates
Stemness kinase
LAG-3
Photosystem (PS)
Adiponectin Receptor
Fas/FasL
PACAP
Anion Exchanger
Thioredoxin
Mucin
Glutathione reductase
MRGPR
Early 2 Factor (E2F)
E3 Ligase Ligand-Linker Conjugates
CPT
CD74
GluCls
NEDD4-1
Cuproptosis
REV-ERB
Fer/FerT kinase
Tight Junction Protein
Lysosomal Autophagy
Glyoxalase
Sodium-dependent phosphate transporter
Poly(ADP-ribose) Glycohydrolase (PARG)
PGC-1α
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