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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
Antibiotic
COX
PI3K
Parasite
AChR
EGFR
Adrenergic Receptor
Ras
HIV Protease
Calcium Channel
Dopamine Receptor
VEGFR
PDE
Dehydrogenase
ROS
Potassium Channel
Cytochromes P450
Epigenetic Reader Domain
Histamine Receptor
Sodium Channel
Histone Methyltransferase
p38 MAPK
HDAC
Antifungal
Phosphatase
ERK
Akt
mTOR
Virus Protease
JAK
SARS-CoV
Src
FLT
Microtubule Associated
Cholinesterase (ChE)
Wnt/beta-catenin
Influenza Virus
STAT
TNF
PARP
iGluR
PDGFR
Reactive Oxygen Species
TRP/TRPV Channel
Topoisomerase
Prostaglandin Receptor
FGFR
GSK-3
Caspase
PKC
Raf
Interleukin
Bcl-2 Family
NO Synthase
HCV Protease
c-Kit
Monoamine Oxidase
GABA Receptor
MMP
Proteasome
c-Met/HGFR
RAAS
MAO
Lipoxygenase
Bcr-Abl
Ferroptosis
JNK
TGF-beta/Smad
ALK
MAPK
HSP
Phospholipase
Transferase
Adenosine Receptor
NMDAR
E1/E2/E3 Enzyme
DUB
Histone Demethylase
GluR
PPAR
Drug Metabolite
Beta Amyloid
Tyrosinase
GPCR
Serine Protease
Aurora Kinase
Integrin
ROCK
Reductase
Kras
Anti-infection
HIF/HIF Prolyl-Hydroxylase
Tyrosine Kinases
Serotonin Transporter
Mitochondrial Metabolism
Casein Kinase
AMPK
PKA
CCR
MDM-2/p53
MEK
ATPase
Serine/threonin kinase
IκB/IKK
HSV
IL Receptor
Reverse Transcriptase
Carbonic Anhydrase
Mitophagy
Nucleoside Antimetabolite/Analog
Angiotensin-converting Enzyme (ACE)
P-gp
Estrogen Receptor/ERR
HBV
IGF-1R
Androgen Receptor
Antiviral
Cysteine Protease
Sirtuin
Glucosidase
CXCR
TLR
Proton pump
RIP kinase
Histone Acetyltransferase
Antioxidant
c-RET
DNA-PK
glycosidase
CaMK
Acyltransferase
TAM Receptor
S6 Kinase
FAK
Leukotriene Receptor
Norepinephrine
NOD-like Receptor (NLR)
LPL Receptor
PERK
c-Fms
HIF
NOS
Estrogen/progestogen Receptor
Gamma-secretase
P2X Receptor
Trk receptor
ATM/ATR
Cannabinoid Receptor
FAAH
Nrf2
NADPH
Opioid Receptor
Hedgehog/Smoothened
Chk
Immunology/Inflammation related
DPP-4
Fatty Acid Synthase
PLK
Kinesin
HER
Neurokinin receptor
Syk
Pim
IDO
Glucocorticoid Receptor
Indoleamine 2,3-Dioxygenase (IDO)
p53
DYRK
Lipase
NOD
HMG-CoA Reductase
Endothelin Receptor
DNA Methyltransferase
PD-1/PD-L1
Chloride channel
Glutathione Peroxidase
Antifection
transporter
PDK
Smo
SGLT
Aryl Hydrocarbon Receptor
Xanthine Oxidase
Hydroxylase
IRAK
LTR
Rho
MAGL
LRRK2
Sigma receptor
Thrombin
ROS Kinase
YAP
P2Y Receptor
c-Myc
BTK
Isocitrate Dehydrogenase (IDH)
PAK
DHFR
Factor Xa
Glutaminase
Stearoyl-CoA Desaturase (SCD)
PGE Synthase
S1P Receptor
Mdm2
Amino Acids and Derivatives
BACE
IAP
Myosin
cAMP
Retinoid Receptor
MRP
Cholecystokinin Receptor
Antifolate
OX Receptor
Epoxide Hydrolase
Beta-Secretase
Aminopeptidase
PI4K
Glucokinase
IRE1
LPA Receptor
Complement System
Monocarboxylate transporter
CSF-1R
Monoamine Transporter
Neuropeptide Y Receptor
OXPHOS
Ephrin Receptor
RSV
ribosome
GTPase
Telomerase
Lipid
PAI-1
Aromatase
AhR
Ligands for Target Protein for PROTAC
DNA
BCRP
Survivin
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Dynamin
Tie-2
PAFR
ABC Transporter
GST
Acetyl-CoA Carboxylase
CFTR
MLK
ADC Cytotoxin
MicroRNA
Necroptosis
GRK
Vasopressin Receptor
STING
Platelet aggregation
NADPH-oxidase
MIF
DNA gyrase
Molecular Glues
Bradykinin Receptor
OAT
MNK
Pyroptosis
Neprilysin
Melanocortin Receptor
CRM1
MyD88
Na+/Ca2+ Exchanger
GNRH Receptor
Neurotensin Receptor
LIM Kinase
NAMPT
PYK2
FLAP
UGT
Glucagon Receptor
GlyT
Wee1
Porcupine
Methionine Adenosyltransferase (MAT)
Carboxypeptidase
SGK
p97
Prolyl Endopeptidase (PREP)
SIK
LDL
Phosphorylase
IKZF
PAD
ATP Citrate Lyase
ASK
CRFR
CGRP Receptor
Gap Junction Protein
DAPK
APC/C
MTP
PROTACs
Adenylyl Cyclase
IFNAR
Bcl-6
LDLR
Arp2/3 Complex
DNA Alkylation
PTEN
cGAS
GPX
Ligand for E3 Ligase
Protease
ROR
DNA Alkylator/Crosslinker
Arrestin
Progesterone Receptor
Melatonin Receptor
AAK1
Guanylate cyclase
MELK
Aquaporin
Thyroid hormone receptor(THR)
Melanin-concentrating Hormone Receptor (MCHR)
MALT
NEDD8
DprE1
Succinate Receptor 1 (SUCNR1)
CETP
Galectin
CaSR
ATG
Liver X Receptor
FXR
NR4A
Amylase
MTH1
MT Receptor
HCN Channel
Bombesin Receptor
CD73
Decarboxylase
Hippo pathway
KLF
CRISPR/Cas9
Oxytocin Receptor
FOXO
Adenosine Deaminase
BMI-1
Advanced Glycation End Products
NPC1L1
CD38
ASBT
TOPK
VDAC
Vitamin
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
Hexokinase
ACK1
p62
FKBP
Imidazoline Receptor
PKM
Apelin receptor
CAT
Transaminase
Arginase
Factor VIIa
ASCT
Hck
Endonuclease
FABP
Haspin Kinase
Somatostatin
KSP
Cadherin
Orphan Receptor
GPCR19
AIM2
TSH Receptor
HuR
GHSR
Ferroportin
PGK1
GSNOR
NUDIX hydrolase
EBI2/GPR183
Y Box Binding Protein 1
Glutaminyl Cyclase
gp120/CD4
Kisspeptin
Photosensitizer
RANKL/RANK
Annexin A
Neuropeptide FF Receptor
Integrase
Transketolase
Huntingtin
PSMA
Urea Transporter
hCE
PARG（Poly(ADP-ribose) Glycohydrolase）
Drug-Linker Conjugates for ADC
FOXO3
Taste receptor
stilbene oxidase
RAR/RXR
Piezo Channel
Procollagen C Proteinase
Aconitase
Neuropeptide W
Cell wall
LHRH
VDA
OCT
N-Acetylglucosaminyltransferase
Stemness kinase
LAG-3
Photosystem (PS)
Adiponectin Receptor
Fas/FasL
PACAP
Anion Exchanger
PROTAC Linker
Thioredoxin
Mucin
Target Protein Ligand-Linker Conjugate
Glutathione reductase
MRGPR
Early 2 Factor (E2F)
CD74
CPT
GluCls
NEDD4-1
Cuproptosis
REV-ERB
Fer/FerT kinase
Tight Junction Protein
Lysosomal Autophagy
Glyoxalase
Sodium-dependent phosphate transporter
Poly(ADP-ribose) Glycohydrolase (PARG)
PGC-1α
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