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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

size

  • 1 mg
  • 10 µL x 10 mM (in DMSO)
  • 20 µL x 10 mM (in DMSO)
  • 30 µL x 10 mM (in DMSO)
  • 50 µL x 10 mM (in DMSO)
  • 100 µL x 10 mM (in DMSO)
  • 250 µL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
Endogenous Metabolite
DNA/RNA Synthesis
NF-κB
CDK
Antibiotic
COX
PI3K
Parasite
Adrenergic Receptor
EGFR
Ras
Calcium Channel
HIV Protease
AChR
Dopamine Receptor
VEGFR
PDE
Dehydrogenase
ROS
Potassium Channel
Cytochromes P450
Histamine Receptor
Epigenetic Reader Domain
Sodium Channel
Histone Methyltransferase
p38 MAPK
ERK
Phosphatase
HDAC
Akt
Antifungal
mTOR
JAK
Virus Protease
SARS-CoV
Src
FLT
Microtubule Associated
Cholinesterase (ChE)
Wnt/beta-catenin
STAT
Influenza Virus
iGluR
PARP
Reactive Oxygen Species
TNF
PDGFR
TRP/TRPV Channel
Topoisomerase
Prostaglandin Receptor
Caspase
GSK-3
FGFR
Interleukin
Raf
PKC
NO Synthase
Bcl-2 Family
HCV Protease
c-Kit
Monoamine Oxidase
GABA Receptor
Proteasome
MMP
c-Met/HGFR
RAAS
JNK
Lipoxygenase
Bcr-Abl
Ferroptosis
ALK
MAO
TGF-beta/Smad
HSP
Phospholipase
MAPK
Transferase
E1/E2/E3 Enzyme
NMDAR
Adenosine Receptor
DUB
GluR
PPAR
Histone Demethylase
Drug Metabolite
BTK
Tyrosinase
Beta Amyloid
Aurora Kinase
Serine Protease
GPCR
Integrin
ROCK
Kras
HIF/HIF Prolyl-Hydroxylase
MDM-2/p53
Casein Kinase
Reductase
PKA
Serotonin Transporter
AMPK
Tyrosine Kinases
CCR
Anti-infection
MEK
Mitochondrial Metabolism
IL Receptor
HSV
Serine/threonin kinase
IκB/IKK
ATPase
Reverse Transcriptase
Carbonic Anhydrase
Nucleoside Antimetabolite/Analog
P-gp
Mitophagy
Angiotensin-converting Enzyme (ACE)
HBV
IGF-1R
Estrogen Receptor/ERR
Antiviral
Androgen Receptor
Sirtuin
Cysteine Protease
TLR
Glucosidase
CXCR
RIP kinase
Histone Acetyltransferase
Antioxidant
Acyltransferase
c-RET
glycosidase
Proton pump
DNA-PK
CaMK
TAM Receptor
FAK
Leukotriene Receptor
Gamma-secretase
S6 Kinase
NOD-like Receptor (NLR)
P2X Receptor
NOS
Norepinephrine
Trk receptor
c-Fms
LPL Receptor
HIF
Estrogen/progestogen Receptor
PERK
ATM/ATR
FAAH
Nrf2
Cannabinoid Receptor
Hedgehog/Smoothened
NADPH
Chk
PLK
Opioid Receptor
Glucocorticoid Receptor
HER
Immunology/Inflammation related
DPP-4
Kinesin
p53
Neurokinin receptor
Pim
IDO
Syk
Fatty Acid Synthase
Indoleamine 2,3-Dioxygenase (IDO)
Lipase
HMG-CoA Reductase
DYRK
NOD
Endothelin Receptor
PD-1/PD-L1
Chloride channel
Glutathione Peroxidase
Xanthine Oxidase
transporter
PDK
DNA Methyltransferase
Antifection
Smo
SGLT
Hydroxylase
Aryl Hydrocarbon Receptor
Sigma receptor
Rho
IRAK
LTR
MAGL
LRRK2
Thrombin
ROS Kinase
YAP
P2Y Receptor
S1P Receptor
Glutaminase
Mdm2
Isocitrate Dehydrogenase (IDH)
PAK
IAP
DHFR
Stearoyl-CoA Desaturase (SCD)
PGE Synthase
Factor Xa
c-Myc
Retinoid Receptor
Amino Acids and Derivatives
cAMP
Epoxide Hydrolase
Cholecystokinin Receptor
Myosin
Beta-Secretase
BACE
PI4K
MRP
Antifolate
Aminopeptidase
IRE1
LPA Receptor
Glucokinase
Complement System
OX Receptor
Monocarboxylate transporter
OXPHOS
CSF-1R
Neuropeptide Y Receptor
RSV
Ephrin Receptor
Monoamine Transporter
ribosome
Telomerase
AhR
GTPase
PAI-1
DNA
Lipid
Ligands for Target Protein for PROTAC
PAFR
BCRP
Survivin
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Aromatase
ABC Transporter
MLK
Tie-2
CFTR
Dynamin
Adenylate cyclase
GST
ADC Cytotoxin
MTP
STING
Acetyl-CoA Carboxylase
NADPH-oxidase
Necroptosis
GRK
MicroRNA
Vasopressin Receptor
Platelet aggregation
DNA gyrase
Bradykinin Receptor
Pyroptosis
Neprilysin
Molecular Glues
OAT
MNK
MIF
ATP Citrate Lyase
Porcupine
MyD88
FLAP
SGK
Glucagon Receptor
CRM1
Neurotensin Receptor
PYK2
UGT
GlyT
Wee1
Methionine Adenosyltransferase (MAT)
p97
Na+/Ca2+ Exchanger
GNRH Receptor
NAMPT
Carboxypeptidase
Melanocortin Receptor
CGRP Receptor
SIK
IKZF
APC/C
Phosphorylase
LIM Kinase
PAD
ASK
DAPK
CRFR
Gap Junction Protein
PROTACs
cGAS
Prolyl Endopeptidase (PREP)
LDL
PTEN
GPX
LDLR
DNA Alkylation
IFNAR
Bcl-6
Arp2/3 Complex
Protease
Ligands for E3 Ligase
Hippo pathway
Arrestin
Melatonin Receptor
Guanylate cyclase
ROR
Aquaporin
Progesterone Receptor
MELK
FOXO
NEDD8
ATG
NR4A
CD73
CRISPR/Cas9
MALT
DprE1
DNA Alkylator/Crosslinker
FXR
Amylase
Thyroid hormone receptor(THR)
Succinate Receptor 1 (SUCNR1)
AAK1
Decarboxylase
Adenosine Deaminase
CETP
MT Receptor
Bombesin Receptor
Galectin
MTH1
KLF
BMI-1
CaSR
Liver X Receptor
HCN Channel
CD38
VDAC
Vitamin
p62
FKBP
Melanin-concentrating Hormone Receptor (MCHR)
NPC1L1
TOPK
Advanced Glycation End Products
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
ACK1
Imidazoline Receptor
Hexokinase
Orphan Receptor
PKM
ASBT
Oxytocin Receptor
Factor VIIa
Endonuclease
PROTAC Linker
TSH Receptor
FABP
KSP
Cadherin
Hck
HuR
Apelin receptor
Haspin Kinase
GPCR19
Transaminase
Somatostatin
CAT
Arginase
ASCT
AIM2
GHSR
PGK1
Ferroportin
PGC-1α
Transketolase
Huntingtin
Kisspeptin
Neuropeptide FF Receptor
Integrase
NUDIX hydrolase
RANKL/RANK
Annexin A
PSMA
hCE
Glutaminyl Cyclase
Urea Transporter
GSNOR
EBI2/GPR183
Y Box Binding Protein 1
gp120/CD4
Photosensitizer
PARG（Poly(ADP-ribose) Glycohydrolase）
Drug-Linker Conjugates for ADC
stilbene oxidase
VDA
N-Acetylglucosaminyltransferase
Target Protein Ligand-Linker Conjugates
LAG-3
Photosystem (PS)
Adiponectin Receptor
Anion Exchanger
E3 Ligase Ligand-Linker Conjugates
CD74
RAR/RXR
Neuropeptide W
PACAP
MRGPR
GluCls
Taste receptor
Aconitase
Thioredoxin
Glutathione reductase
Piezo Channel
Procollagen C Proteinase
Cell wall
OCT
Stemness kinase
Fas/FasL
Early 2 Factor (E2F)
FOXO3
NEDD4-1
Fer/FerT kinase
Tight Junction Protein
Glyoxalase
Mucin
Cuproptosis
LHRH
CPT
REV-ERB
Lysosomal Autophagy
Sodium-dependent phosphate transporter
Poly(ADP-ribose) Glycohydrolase (PARG)
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