Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Mesembrine ((+)-Mesembrine), a primary alkaloid distinguished by its aryloctahydroindole structure, acts as a potent 5-HT transporter inhibitor with an inhibition constant (K i) of 1.4 nM. Additionally, it demonstrates inhibitory activity against phosphodiesterase 4B (PDE4B) with an inhibitory concentration 50% (IC50) of 7.8 μM [1] [2].
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Description | Mesembrine ((+)-Mesembrine), a primary alkaloid distinguished by its aryloctahydroindole structure, acts as a potent 5-HT transporter inhibitor with an inhibition constant (K i) of 1.4 nM. Additionally, it demonstrates inhibitory activity against phosphodiesterase 4B (PDE4B) with an inhibitory concentration 50% (IC50) of 7.8 μM [1] [2]. |
Molecular Weight | 289.37 |
Formula | C17H23NO3 |
CAS No. | 468-53-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Mesembrine 468-53-1 inhibitor inhibit