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Dazcapistat

Name: Dazcapistat
Brand: TargetMol
SKU: T9710
Price: 88 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T9710Cas No. 2221010-42-8

Dazcapistat is a potent calpain inhibitor with IC50s of <3 μM for calpain 1, calpain 2, and calpain 9, respectively.

Dazcapistat

🥰Excellent

Purity: 99.11%

Catalog No. T9710Cas No. 2221010-42-8

Dazcapistat is a potent calpain inhibitor with IC50s of <3 μM for calpain 1, calpain 2, and calpain 9, respectively.

Pack Size	Price	Availability
1 mg	$88	In Stock
5 mg	$213	In Stock
10 mg	$322	In Stock
25 mg	$579	In Stock
50 mg	$813	In Stock
100 mg	$1,130	In Stock
1 mL x 10 mM (in DMSO)	$235	In Stock

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Batch Information

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Purity:99.11%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	Dazcapistat is a potent calpain inhibitor with IC50s of <3 μM for calpain 1, calpain 2, and calpain 9, respectively.
Targets&IC50	Calpain:<3 μM

Chemical Properties

Molecular Weight	395.38
Formula	C₂₁H₁₈FN₃O₄
Cas No.	2221010-42-8
Smiles	Cc1nc(c(o1)C(=O)NC(Cc1ccccc1)C(=O)C(N)=O)-c1ccccc1F
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 45 mg/mL (113.81 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.5292 mL	12.6461 mL	25.2921 mL	126.4606 mL
5 mM	0.5058 mL	2.5292 mL	5.0584 mL	25.2921 mL
10 mM	0.2529 mL	1.2646 mL	2.5292 mL	12.6461 mL
20 mM	0.1265 mL	0.6323 mL	1.2646 mL	6.3230 mL
50 mM	0.0506 mL	0.2529 mL	0.5058 mL	2.5292 mL
100 mM	0.0253 mL	0.1265 mL	0.2529 mL	1.2646 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc