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Sodium Channel inhibitor 4

Name: Sodium Channel inhibitor 4
Brand: TargetMol
SKU: T81134
Price: 40 USD
Availability: InStock
Rating: 5 (10 reviews)

Catalog No. T81134 Copy Product Info

Purity: 99.89%

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Sodium Channel inhibitor 4 is a potent and selective NaV1.7 inhibitor (IC50 = 33 nM). It blocks action potential conduction in sensory neurons, exhibiting significant analgesic activity for neuropathic pain research.

Sodium Channel inhibitor 4

Copy Product Info

🥰Excellent

Catalog No. T81134

Cas No. 587843-16-1

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Pack Size	Price	USA Stock	Global Stock
5 mg	$40	-	In Stock
10 mg	$64	-	In Stock
25 mg	$106	-	In Stock
50 mg	$155	-	In Stock

For In stock only · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)

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For research use only—not for human use. No sales to individuals. Use as intended only.

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Batch Information

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Purity:99.89%

Appearance:Solid

Color:White

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description

Chemical Properties

Molecular Weight	451.95
Formula	C₁₉H₁₈ClN₃O₄S₂
Cas No.	587843-16-1
Smiles	O=C(NC1=CC=C(C=C1)S(=O)(=O)NC2=NC=CS2)C(OC3=CC=C(Cl)C=C3)(C)C

Storage & Solubility Information

Storage

keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 80 mg/mL (177.01 mM), Sonication is recommmended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.2126 mL	11.0632 mL	22.1263 mL	110.6317 mL
5 mM	0.4425 mL	2.2126 mL	4.4253 mL	22.1263 mL
10 mM	0.2213 mL	1.1063 mL	2.2126 mL	11.0632 mL
20 mM	0.1106 mL	0.5532 mL	1.1063 mL	5.5316 mL
50 mM	0.0443 mL	0.2213 mL	0.4425 mL	2.2126 mL
100 mM	0.0221 mL	0.1106 mL	0.2213 mL	1.1063 mL

Note : The dilution table applies only to solid products. For liquid products, please calculate the stock solution based on the stated concentration and/or density.

Calculator

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc