Shopping Cart

Remove All
Your shopping cart is currently empty

Pinacidil monohydrate

Name: Pinacidil monohydrate
Brand: TargetMol
SKU: T12478
Price: 29 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T12478Cas No. 85371-64-8

Pinacidil monohydrate is a potassium channel activator, antihypertensive drug.

Pinacidil monohydrate

🥰Excellent

Purity: 99.98%

Catalog No. T12478Cas No. 85371-64-8

Pinacidil monohydrate is a potassium channel activator, antihypertensive drug.

Pack Size	Price	Availability
10 mg	$29	In Stock
25 mg	$48	In Stock
50 mg	$77	In Stock
1 mL x 10 mM (in DMSO)	$29	In Stock

Add to Cart

Add to Quotation

Bulk & Custom

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

Select Batch

Purity:99.98%

Resource Download

COA HNMR LCMS HPLC

Product Introduction

Bioactivity

Description	Pinacidil monohydrate is a potassium channel activator, antihypertensive drug.
In vitro	Pinacidil hydrate activates the ATP-modulated potassium channels of guinea pog bladder and heart with Ki values of 104 and 251 nM, respectively[3].

Chemical Properties

Molecular Weight	263.34
Formula	C₁₃H₂₁N₅O
Cas No.	85371-64-8
Smiles	O.CC(N\C(Nc1ccncc1)=N/C#N)C(C)(C)C
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 97 mg/mL (368.35 mM), Sonication is recommended.

Ethanol: 47 mg/mL (178.48 mM), Sonication is recommended.

Solution Preparation Table

Ethanol/DMSO

	1mg	5mg	10mg	50mg
1 mM	3.7974 mL	18.9869 mL	37.9737 mL	189.8686 mL
5 mM	0.7595 mL	3.7974 mL	7.5947 mL	37.9737 mL
10 mM	0.3797 mL	1.8987 mL	3.7974 mL	18.9869 mL
20 mM	0.1899 mL	0.9493 mL	1.8987 mL	9.4934 mL
50 mM	0.0759 mL	0.3797 mL	0.7595 mL	3.7974 mL
100 mM	0.0380 mL	0.1899 mL	0.3797 mL	1.8987 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc