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FATP1-IN-2

Name: FATP1-IN-2
Brand: TargetMol
SKU: T40287
Price: 499 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T40287Cas No. 2650944-83-3

FATP1-IN-2 is a fatty acid transporter protein 1 (FATP1) inhibitor with oral activity for the study of obesity and metabolic diseases.

FATP1-IN-2

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Purity: 98.49%

Catalog No. T40287Cas No. 2650944-83-3

FATP1-IN-2 is a fatty acid transporter protein 1 (FATP1) inhibitor with oral activity for the study of obesity and metabolic diseases.

Pack Size	Price	USA Warehouse	Global Warehouse	Quantity
2 mg	$499	-	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Batch Information

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Purity:98.49%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	FATP1-IN-2 is a fatty acid transporter protein 1 (FATP1) inhibitor with oral activity for the study of obesity and metabolic diseases.
Targets&IC50	FATP1 (human):0.43 μM, FATP1 (mouse):0.39 μM
In vivo	FATP1-IN-2 (10 mg/kg; oral; Mice) showed a Cmax value above the mouse IC50 value.[1] FATP1-IN-2 (3, 10, 30 mg/kg; oral; for 4 weeks; Mice) showed no change in the TG content of each tissue at any dose.[1]

Chemical Properties

Molecular Weight	353.39
Formula	C₁₉H₂₀FN₅O
Cas No.	2650944-83-3
Smiles	Cc1nc2ccccn2c1C(=O)CN1CCN(CC1)c1ccc(F)cn1

Storage & Solubility Information

Storage

store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 80 mg/mL (226.38 mM), Sonication is recommended.

In Vivo Formulation

10% DMSO+40% PEG300+5% Tween 80+45% Saline: 5 mg/mL (14.15 mM), Sonication is recommended.

Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.8297 mL	14.1487 mL	28.2973 mL	141.4867 mL
5 mM	0.5659 mL	2.8297 mL	5.6595 mL	28.2973 mL
10 mM	0.2830 mL	1.4149 mL	2.8297 mL	14.1487 mL
20 mM	0.1415 mL	0.7074 mL	1.4149 mL	7.0743 mL
50 mM	0.0566 mL	0.2830 mL	0.5659 mL	2.8297 mL
100 mM	0.0283 mL	0.1415 mL	0.2830 mL	1.4149 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline /PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline /PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

FATP1-IN-2FATP-1-IN-2FATP1IN2FATP1 IN 2FATP