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Acetyl-Calpastatin (184-210)(human) acetate

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TargetMol
Catalog No. TP2056L
Alias Acetyl-Calpastatin (184-210) (human) acetate(123714-50-1 Free base )

Acetyl-Calpastatin (184-210)(human) acetate is a potent, selective and reversible calpain inhibitor with Ki values of 0.2 nM and 6 μM for µ-calpain and cathepsin L, respectively.

Acetyl-Calpastatin (184-210)(human) acetate
Other Forms of Acetyl-Calpastatin (184-210)(human) acetate:
Acetyl-Calpastatin(184-210)(human)TP2056123714-50-1
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Acetyl-Calpastatin (184-210)(human) acetate

🥰Excellent
TargetMol
Purity: 98.16%
Catalog No. TP2056LAlias Acetyl-Calpastatin (184-210) (human) acetate(123714-50-1 Free base )
Acetyl-Calpastatin (184-210)(human) acetate is a potent, selective and reversible calpain inhibitor with Ki values of 0.2 nM and 6 μM for µ-calpain and cathepsin L, respectively.
Pack SizePriceAvailabilityQuantity
1 mg$117In Stock
5 mg$269In Stock
10 mg$395In Stock
25 mg$592In Stock
50 mg$833In Stock
100 mg$1,120In Stock
200 mg$1,520In Stock
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Purity:98.16%
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COA HPLC MS

Product Introduction

Bioactivity
Description
Acetyl-Calpastatin (184-210)(human) acetate is a potent, selective and reversible calpain inhibitor with Ki values of 0.2 nM and 6 μM for µ-calpain and cathepsin L, respectively.
In vitro
Acetyl-Calpastatin (184-210)(human) acetate (peptide 1; 12.5-100 μM) inhibits calpains in LCLC 103H cells with an IC50 of 27 μM[1].
SynonymsAcetyl-Calpastatin (184-210) (human) acetate(123714-50-1 Free base )
Chemical Properties
Molecular Weight3237.68
FormulaC144H234N36O46S
SmilesCC(O)=O.CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CO)NC(=O)[C@H](CCSC)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CC(O)=O)NC(C)=O)[C@@H](C)O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(N)=O
SequenceAc-Asp-Pro-Met-Ser-Ser-Thr-Tyr-Ile-Glu-Glu-Leu-Gly-Lys-Arg-Glu-Val-Thr-Ile-Pro-Pro-Lys-Tyr-Arg-Glu-Leu-Leu-Ala-NH2
Sequence ShortAc-DPMSSTYIEELGKREVTIPPKYRELLA-NH2
Storage & Solubility Information
Storagestore at low temperature,keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
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Keywords

CysteineProteaseCysteine ProteaseCalpainAcetyl-Calpastatin AcetateAcetyl-Calpastatin
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