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BEBT-908

Name: BEBT-908
Brand: TargetMol
SKU: T16529
Price: 117 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T16529Cas No. 1235449-52-1

Alias PI3Kα inhibitor 1, MDK9521

BEBT-908 (PI3Kα inhibitor 1) is a selective PI3Kα inhibitor with an IC50 of less than 0.1 μM and also inhibits HDAC with an IC50 ranging from 0.1 μM to 1 μM.

BEBT-908

🥰Excellent

Purity: 99.67%

Catalog No. T16529Alias PI3Kα inhibitor 1, MDK9521Cas No. 1235449-52-1

BEBT-908 (PI3Kα inhibitor 1) is a selective PI3Kα inhibitor with an IC50 of less than 0.1 μM and also inhibits HDAC with an IC50 ranging from 0.1 μM to 1 μM.

Pack Size	Price	Availability
1 mg	$117	In Stock
5 mg	$250	In Stock
10 mg	$377	In Stock
25 mg	$630	In Stock
50 mg	$898	In Stock
100 mg	$1,210	In Stock
200 mg	$1,630	In Stock
1 mL x 10 mM (in DMSO)	$278	In Stock

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Batch Information

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Purity:99.67%

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description	BEBT-908 (PI3Kα inhibitor 1) is a selective PI3Kα inhibitor with an IC50 of less than 0.1 μM and also inhibits HDAC with an IC50 ranging from 0.1 μM to 1 μM.
Targets&IC50	HDAC:0.1 μM, PI3Kα:0.1 μM
Alias	PI3Kα inhibitor 1, MDK9521

Chemical Properties

Molecular Weight	507.57
Formula	C₂₃H₂₅N₉O₃S
Cas No.	1235449-52-1
Smiles	CNc1ccc(cn1)-c1nc(N2CCOCC2)c2sc(CN(C)c3ncc(cn3)C(=O)NO)cc2n1
Relative Density.	1.461 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 35 mg/mL (68.96 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.9702 mL	9.8509 mL	19.7017 mL	98.5086 mL
5 mM	0.3940 mL	1.9702 mL	3.9403 mL	19.7017 mL
10 mM	0.1970 mL	0.9851 mL	1.9702 mL	9.8509 mL
20 mM	0.0985 mL	0.4925 mL	0.9851 mL	4.9254 mL
50 mM	0.0394 mL	0.1970 mL	0.3940 mL	1.9702 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc