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ALR2-IN-1

Name: ALR2-IN-1
Brand: TargetMol
SKU: T77523
Price: 32 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T77523Cas No. 2799695-54-6

ALR2-IN-1 is a potent and selective ALR2 inhibitor with an IC50 value of 1.42 μM. ALR2-IN-1 possesses both antiglycemic and antioxidant activities and can be used to study the complications of diabetes.

ALR2-IN-1

🥰Excellent

Purity: 98.79%

Catalog No. T77523Cas No. 2799695-54-6

Pack Size	Price	Availability
5 mg	$32	In Stock
10 mg	$56	In Stock
25 mg	$119	In Stock
50 mg	$191	In Stock
100 mg	$286	In Stock
200 mg	$405	In Stock

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Batch Information

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Purity:98.79%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	ALR2-IN-1 is a potent and selective ALR2 inhibitor with an IC50 value of 1.42 μM. ALR2-IN-1 possesses both antiglycemic and antioxidant activities and can be used to study the complications of diabetes.
Targets&IC50	ALR2:1.42 μM

Chemical Properties

Molecular Weight	315.39
Formula	C₁₆H₁₇N₃O₂S
Cas No.	2799695-54-6
Smiles	N(C(NN=CC1=C(O)C=CC(C)=C1)=S)C2=CC(OC)=CC=C2
Relative Density.	1.22 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 90.0 mg/mL (285.4 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.1707 mL	15.8534 mL	31.7068 mL	158.5339 mL
5 mM	0.6341 mL	3.1707 mL	6.3414 mL	31.7068 mL
10 mM	0.3171 mL	1.5853 mL	3.1707 mL	15.8534 mL
20 mM	0.1585 mL	0.7927 mL	1.5853 mL	7.9267 mL
50 mM	0.0634 mL	0.3171 mL	0.6341 mL	3.1707 mL
100 mM	0.0317 mL	0.1585 mL	0.3171 mL	1.5853 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc