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TargetMol | Compound Library

FDA-Approved Kinase Inhibitor Library

Catalog No. L1610

Kinases are a class of enzymes that facilitates phosphorylation, by transferring phosphate groups from high-energy donor molecules, such as ATP, to specific target molecules. A common group of kinases are the protein kinases, which act on specific proteins to phosphorylate them and alter their activity. Protein kinases are involved in a range of cell signaling and regulatory processes and play an important role in cell growth, metabolism, differentiation and apoptosis. Protein kinases have been associated with many diseases, including cancer, inflammatory diseases, cardiovascular diseases and neurological disorders. Therefore, targeting protein kinases has emerged as a promising therapeutic strategy for the treatment of related diseases. Targetmol's FDA-Approved Kinase Inhibitor Library contains 263 marketed drugs that target kinases. These kinases include Insulin/IGF Receptors,PI 3-Kinase,CaM Kinase II,JAK,PKA,CDK,JNK,PKC,CKI II,MAPK,RAF,EGFR,MEK,SAPK,GSK,MLCK,Src-family,IKK,PDGFR,VEGFR etc. FDA-Approved Kinase Inhibitor Library is a powerful tool for kinase drug development and related research.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L1610

FDA-Approved Kinase Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 263 kinase inhibitors/regulators for specific targeting of kinases, ready for high-throughput screening and high-content screening.
  • All compounds have undergone preclinical studies and clinical trials, approved for marketing by FDA, EMA, PMDA, etc., with proven biological activity and safety.
  • Detailed instructions, compound structures, target information, IC50 values, activity descriptions, etc.
  • NMR, HPLC/LCMS and other assay techniques to ensure the correct structure and high purity of the product and reduce false positives.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
EGFR
VEGFR
c-Kit
PDGFR
FGFR
JAK
FLT
Src
Bcr-Abl
c-Met/HGFR
Tyrosine Kinases
ALK
PKC
CDK
Raf
Endogenous Metabolite
Mitophagy
NF-κB
AMPK
Antibacterial
c-RET
Adrenergic Receptor
Antibiotic
CaMK
PI3K
ROCK
Sodium Channel
5-HT Receptor
Ferroptosis
MEK
mTOR
PKA
Potassium Channel
Trk receptor
Calcium Channel
HER
Parasite
ROS Kinase
TAM Receptor
AChR
Akt
COX
ERK
Histamine Receptor
HIV Protease
PDE
ROS
Antifungal
Dopamine Receptor
GSK-3
Influenza Virus
IκB/IKK
p38 MAPK
c-Fms
Cytochromes P450
FAK
Glucosidase
IGF-1R
Microtubule Associated
NADPH
Nrf2
PAK
Serine/threonin kinase
Syk
Topoisomerase
BTK
Adenosine Receptor
Aurora Kinase
Dehydrogenase
DNA/RNA Synthesis
Ephrin Receptor
Glutathione Peroxidase
Hexokinase
Interleukin
IRE1
Kras
Ligands for Target Protein for PROTAC
Lipoxygenase
LPL Receptor
MAPK
P-gp
Ras
ROR
S1P Receptor
SARS-CoV
Serotonin Transporter
TNF
TOPK
ACK1
Antifolate
Anti-infection
Antioxidant
Antiviral
ATP Citrate Lyase
Beta Amyloid
Caspase
Chk
Chloride channel
Cholinesterase (ChE)
CSF-1R
DHFR
DNA
DNA-PK
Estrogen/progestogen Receptor
Gap Junction Protein
Glucokinase
GluR
gp120/CD4
GRK
HBV
Hck
HCV Protease
HDAC
HIF/HIF Prolyl-Hydroxylase
HSV
Hydroxylase
IFNAR
IL Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Integrin
JNK
LDL
Melatonin Receptor
Mitochondrial Metabolism
Monoamine Transporter
NADPH-oxidase
NO Synthase
Norepinephrine
Nucleoside Antimetabolite/Analog
PAD
PDK
Phosphatase
PKM
PLK
PPAR
Proton pump
Reactive Oxygen Species
S6 Kinase
Serine Protease
Sigma receptor
Sirtuin
TGF-beta/Smad
Transferase
TRP/TRPV Channel
Tyrosinase
Virus Protease
YAP
ADC Cytotoxin

Keywords