Powder: -20°C for 3 years | In solvent: -80°C for 1 year
MSC2504877 is an inhibitor of tankyrase and enhances the effects of clinical CDK4/6 inhibitors. MSC2504877 suppresses the upregulation of Cyclin D2 and Cyclin E2 caused by palbociclib and enhances the suppression of phospho-Rb.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 67.00 | |
5 mg | In stock | $ 153.00 | |
10 mg | In stock | $ 243.00 | |
25 mg | In stock | $ 473.00 | |
50 mg | In stock | $ 693.00 | |
100 mg | In stock | $ 988.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 153.00 |
Description | MSC2504877 is an inhibitor of tankyrase and enhances the effects of clinical CDK4/6 inhibitors. MSC2504877 suppresses the upregulation of Cyclin D2 and Cyclin E2 caused by palbociclib and enhances the suppression of phospho-Rb. |
Synonyms | 3-(4-(2-Hydroxypropan-2-yl)phenyl)-6-methylpyrrolo[1,2-a]pyrazin-1(2H)-one |
Molecular Weight | 282.34 |
Formula | C17H18N2O2 |
CAS No. | 1460286-21-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 3.6 mg/mL (12.75 mM)
You can also refer to dose conversion for different animals. More
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MSC2504877 1460286-21-8 Others MSC-2504877 3-(4-(2-Hydroxypropan-2-yl)phenyl)-6-methylpyrrolo[1,2-a]pyrazin-1(2H)-one MSC 2504877 inhibitor inhibit