store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
MRTX0902 is an effective and high selective inhibitor of SOS1 with an IC50 of 46 nM and a Ki of 2 nM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 87.00 | |
5 mg | In stock | $ 213.00 | |
10 mg | In stock | $ 313.00 | |
25 mg | In stock | $ 663.00 | |
50 mg | In stock | $ 1,060.00 | |
100 mg | In stock | $ 1,730.00 |
Description | MRTX0902 is an effective and high selective inhibitor of SOS1 with an IC50 of 46 nM and a Ki of 2 nM. |
In vitro | In the MIA PaCa-2 xenograft model of mice, MRTX0902 (25 and 50 mg/kg; p.o.) shows anti-tumor effects and reduces tumor growth by 41% and 53%, respectively[1]. |
Synonyms | UNII-CRG69FR93G |
Molecular Weight | 388.47 |
Formula | C22H24N6O |
CAS No. | 2654743-22-1 |
store at low temperature
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 10 mg/mL (25.7 mM), Sonication and heating to 60℃ are recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
MRTX0902 2654743-22-1 MAPK Raf UNII-CRG69FR93G MRTX 0902 MRTX-0902 inhibitor inhibit