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PD 117519

🥰Excellent
Catalog No. T7509Cas No. 96392-15-3
Alias CI947

PD 117519 (CI947) is an agonist of the adenosine receptor.

PD 117519

PD 117519

🥰Excellent
Purity: 99.98%
Catalog No. T7509Alias CI947Cas No. 96392-15-3
PD 117519 (CI947) is an agonist of the adenosine receptor.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
2 mg$30In StockIn Stock
5 mg$50In StockIn Stock
10 mg$83In StockIn Stock
25 mg$148In StockIn Stock
50 mg$271In StockIn Stock
100 mg$397In StockIn Stock
1 mL x 10 mM (in DMSO)$55In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Batch Information

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Purity:99.98%
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COA HNMR LCMS

Product Introduction

Bioactivity
Description
PD 117519 (CI947) is an agonist of the adenosine receptor.
In vivo
PD 117519?selectively binds to adenosine A2 receptors (IC50 = 30 μM) over A1 receptors (IC50 = 810 μM) in rat brain membranes.?PD 117519 increases heart rate and decreases systolic blood pressure in normotensive dogs when administered at doses of 2 or 10 mg/kg[1].
SynonymsCI947
Chemical Properties
Molecular Weight383.4
FormulaC19H21N5O4
Cas No.96392-15-3
SmilesOC[C@H]1O[C@H]([C@H](O)[C@@H]1O)n1cnc2c(NC3Cc4ccccc4C3)ncnc12
Relative Density.1.71g/cm3
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 100 mg/mL (260.82 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.6082 mL13.0412 mL26.0824 mL130.4121 mL
5 mM0.5216 mL2.6082 mL5.2165 mL26.0824 mL
10 mM0.2608 mL1.3041 mL2.6082 mL13.0412 mL
20 mM0.1304 mL0.6521 mL1.3041 mL6.5206 mL
50 mM0.0522 mL0.2608 mL0.5216 mL2.6082 mL
100 mM0.0261 mL0.1304 mL0.2608 mL1.3041 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
% DMSO
%
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Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

PD-117519PD117519PD 117519P1 receptorInhibitorinhibitCI-947CI 947AdenosineReceptorAdenosine ReceptorA2
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