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Perospirone hydrochloride

Name: Perospirone hydrochloride
Brand: TargetMol
SKU: T8136
Price: 30 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T8136Cas No. 129273-38-7

Alias SM-9018 hydrochloride, Perospirone HCl

Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia. It also displays affinity towards 5HT1A receptors as a partial agonist.

Perospirone hydrochloride

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Purity: 99.37%

Catalog No. T8136Alias SM-9018 hydrochloride, Perospirone HClCas No. 129273-38-7

Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia. It also displays affinity towards 5HT1A receptors as a partial agonist.

Pack Size	Price	USA Warehouse	Global Warehouse
25 mg	$38	In Stock	In Stock
50 mg	$56	In Stock	In Stock
100 mg	$82	In Stock	In Stock
200 mg	$118	-	In Stock
1 mL x 10 mM (in DMSO)	$30	In Stock	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Batch Information

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Purity:99.37%

Appearance:Solid

Color:White

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description	Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia. It also displays affinity towards 5HT1A receptors as a partial agonist.
Targets&IC50	5-HT1 receptor:18 nM (Ki), D1 receptor:41 nM (Ki), 5-HT1A receptor:2.9 nM (Ki), 5-HT2A receptor:0.6 nM (Ki), D2 receptor:1.4 nM (Ki)
Synonyms	SM-9018 hydrochloride, Perospirone HCl

Chemical Properties

Molecular Weight	463
Formula	C₂₃H₃₁ClN₄O₂S
Cas No.	129273-38-7
Smiles	Cl.O=C1C2CCCCC2C(=O)N1CCCCN1CCN(c2nsc3ccccc23)CC1
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 92 mg/mL (198.7 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.1598 mL	10.7991 mL	21.5983 mL	107.9914 mL
5 mM	0.4320 mL	2.1598 mL	4.3197 mL	21.5983 mL
10 mM	0.2160 mL	1.0799 mL	2.1598 mL	10.7991 mL
20 mM	0.1080 mL	0.5400 mL	1.0799 mL	5.3996 mL
50 mM	0.0432 mL	0.2160 mL	0.4320 mL	2.1598 mL
100 mM	0.0216 mL	0.1080 mL	0.2160 mL	1.0799 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc