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Cudetaxestat

Catalog No. T63190 CAS 1782070-21-6

Synonyms: BLD-0409

Cudetaxestat is a potent inhibitor of orally active autotaxin.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Cudetaxestat, CAS 1782070-21-6

Pack Size	Availability	Price/USD
1 mg	In stock	$ 198.00
5 mg	In stock	$ 383.00
10 mg	In stock	$ 617.00
25 mg	In stock	$ 1,219.00
50 mg	In stock	$ 1,967.00
100 mg	In stock	$ 3,155.00
1 mL * 10 mM (in DMSO)	In stock	$ 399.00

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Purity: 98.84%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Cudetaxestat is a potent inhibitor of orally active autotaxin.

Synonyms	BLD-0409
Molecular Weight	482.33
Formula	C21H15Cl2F2N3O2S
CAS No.	1782070-21-6

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 225.0 mg/mL (466.5 mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Tan Z, et al. An updated patent review of autotaxin inhibitors (2017-present). Expert Opin Ther Pat. 2021;31(5):421-434.

Related compound libraries

This product is contained In the following compound libraries：

Inhibitor Library

Related Products

Related compounds with same targets

Pterine-6-carboxylic acid Norbraylin Vardenafil dihydrochloride PF-05180999 PAT-048 K134 PAT-505 OR-1896

Dose Conversion

You can also refer to dose conversion for different animals. More

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Calculation results:

Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

Note:

Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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The answer of 19.713 mg appears in the Mass box

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An example of a dilution calculation using the Tocris dilution calculator
What volume of a given 10 mM stock solution is required to make 20ml of a 50 μM solution?
Using the equation C1V1 = C2V2, where C1=10 mM, C2=50 μM, V2=20 ml and V1 is the unknown:
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The answer of 100 microliter (0.1 ml) appears in the Volume (start) box

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Molar mass (molar weight) is the mass of one mole of a substance and is expressed in g/mol.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Cudetaxestat 1782070-21-6 Metabolism PDE BLD-0409 Inhibitor inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.