TN1033 |
Sennidin A
|
641-12-3
|
100%
|
|
Sennidin A, has two hydroxyanthraquinone-like moieties, exerts inhibition on NS3 helicase with IC50 values of 0.8 μM.
|
TN1034 |
Sennidin B
|
517-44-2
|
|
|
Sennidin B stimulates glucose incorporation in rat adipocytes.
|
TN3885 |
Dodoviscin J
|
1372527-42-8
|
98%
|
|
Dodoviscin J can promote adipocyte differentiation as characterized by increased triglyceride levels in 3T3L1 cells.
|
TN1681 |
Gentianine
|
439-89-4
|
98%
|
|
Gentianine is an effective Swertiamarin derivative, which has anti-diabetic, antipsychotic, anti-inflammatory, hypotensive, diuretic and other effects, and has t...
|
TN3884 |
Dodoviscin I
|
1372527-40-6
|
98%
|
|
Dodoviscin I can promote adipocyte differentiation as characterized by increased triglyceride levels in 3T3L1 cells.
|
TMA0127 |
Ficusin A
|
173429-83-9
|
98%
|
|
Ficusin has antioxidant, antilipidemic and antidiabetic effects, it can lower the levels of fasting blood glucose, plasma insulin, body weight gain in HFD-STZ in...
|
TN3882 |
Dodoviscin A
|
1372527-25-7
|
98%
|
|
Dodoviscin A may be a new promising pigmentation-altering agent for cosmetic and therapeutic applications, it can inhibit melanin biosynthesis induced by 3-isobu...
|
TN2535 |
1-Hydroxy-2-oxopomolic acid
|
217466-37-0
|
98%
|
|
1β-Hydroxy-2-oxopomolic acid inhibits adipocyte differentiation through downregulation of various adipocytokines by blocking PPARγ and C/EBPα expression.
|
T11055 |
DL-TBOA
|
205309-81-5
|
98%
|
|
DL-TBOA inhibited [14C] glutamate uptake in COS-1 cells expressing human EAAT1 and EAAT2, with Ki values of 42 μM and 5.7 μM, respectively. DL-TBOA blocks EAAT4 ...
|
TN3883 |
Dodoviscin H
|
1372527-39-3
|
98%
|
|
Dodoviscin H can promote adipocyte differentiation as characterized by increased triglyceride levels in 3T3L1 cells.
|
T40083 |
GLUT inhibitor-1
|
2421141-40-2
|
98%
|
|
GLUT inhibitor-1 is an orally active GLUT inhibitor with IC50 s of 242 nM and 179 nM for GLUT1 and GLUT3. GLUT inhibitor-1 can be used in studies about cancers a...
|
T13330L |
WAY-213613
|
868359-05-1
|
98%
|
|
WAY-213613 is a potent and selective nonsubstrate reuptake inhibitor of GLT-1/EAAT2 (IC50: 85 nM EAAT2). It displays 59- and 44-fold selectivity over EAAT1 and E...
|
T8616 |
Fasentin
|
392721-37-8
|
99.95%
|
|
Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) is an inhibitor of GluT1.
|
T2363 |
STF-31
|
724741-75-7
|
99.92%
|
|
STF-31 is an inhibitor of glucose transporter 1 (GLUT1) with IC50 of 1 μM.
|
T15446 |
GT 949
|
460330-27-2
|
99.89%
|
|
GT 949 is a selective excitatory positive allosteric modulator of amino acid transporter-2 (EAAT2) (EC50: 0.26 nM).
|
T6797 |
Telaglenastat
|
1439399-58-2
|
99.87%
|
|
Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.
|
T77657 |
MSNBA
|
852702-51-3
|
99.86%
|
|
MSNBA is a selective and potent inhibitor of fructose transport through GLUT5 and also acts as a probe of the GLUT5 transporter. MSNBA inhibited GLUT5 fructose u...
|
TN5137 |
Tetramethylkaempferol
|
16692-52-7
|
99.65%
|
|
Tetramethylkaempferol is a PPARγ agonist, it can improve insulin sensitivity by increasing the levels of adiponectin, an important adipocytokine associated with ...
|
T9347 |
EAAT2 activator 1
|
892415-28-0
|
99.63%
|
|
EAAT2 activator 1 (3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine) is a thiopyridazine derivative that has been found to increase EAAT2 protein level...
|
T9590 |
T-1095
|
209746-59-8
|
99.56%
|
|
T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) and facilitative glucose transporter 2 (GLUT2).
|