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Cenupatide

Name: Cenupatide
Brand: TargetMol
SKU: TP2338
Rating: 4.5 (1 reviews)

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Catalog No. TP2338Cas No. 1006388-38-0

Alias Ac-Arg-Aib-Arg-α(Me)Phe-NH2

Cenupatide is a urokinase plasminogen activator receptor (uPAR) inhibitor. Cenupatide inhibits uPAR binding to the formyl peptide receptors (FPRs) can improve kidney lesions in a rat model of STZ-induced diabetes. Cenupatide reverted STZ-induced up-regulation of uPA levels and activity, while uPAR on podocytes and (s)uPAR were unaffected. In glomeruli, Cenupatide inhibited FPR2 expression.

Cenupatide

😃Good

Catalog No. TP2338Alias Ac-Arg-Aib-Arg-α(Me)Phe-NH2Cas No. 1006388-38-0

Pack Size	Price	Availability
5 mg	$152	Backorder
10 mg	$255	Backorder
25 mg	$461	Backorder
50 mg	$875	Backorder
100 mg	$1,496	Backorder
200 mg	$2,323	Backorder

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Product Introduction

Bioactivity

Description	Cenupatide is a urokinase plasminogen activator receptor (uPAR) inhibitor. Cenupatide inhibits uPAR binding to the formyl peptide receptors (FPRs) can improve kidney lesions in a rat model of STZ-induced diabetes. Cenupatide reverted STZ-induced up-regulation of uPA levels and activity, while uPAR on podocytes and (s)uPAR were unaffected. In glomeruli, Cenupatide inhibited FPR2 expression.
Synonyms	Ac-Arg-Aib-Arg-α(Me)Phe-NH2

Chemical Properties

Molecular Weight	617.756
Formula	C₂₈H₄₇N₁₁O₅
Cas No.	1006388-38-0
Relative Density.	1.34 g/cm3 (Predicted)
Sequence	Ac-Arg-{Aib}-Arg-{aMePhe}-NH2
Sequence Short	Ac-R-{Aib}-R-{aMePhe}-NH2

Storage & Solubility Information

Storage

keep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

Cenupatide trifluoroacetic acidCenupatideAc-Arg-Aib-Arg-α(Me)Phe-NH2)Ac-Arg-Aib-Arg-alpha(Me)Phe-NH2)Ac-Arg-Aib-Arg-a(Me)Phe-NH2)