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Urapidil

Name: Urapidil
Brand: TargetMol
SKU: T0165
Price: 33 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T0165Cas No. 34661-75-1

Alias Mediatensyl, Eupressyl, Ebrantil

Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.

Urapidil

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Purity: 99.85%

Catalog No. T0165Alias Mediatensyl, Eupressyl, EbrantilCas No. 34661-75-1

Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.

Pack Size	Price	Availability
25 mg	$33	In Stock
50 mg	$47	In Stock
100 mg	$68	In Stock
500 mg	$159	In Stock
1 mL x 10 mM (in DMSO)	$39	In Stock

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Batch Information

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Purity:99.85%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
Synonyms	Mediatensyl, Eupressyl, Ebrantil

Chemical Properties

Molecular Weight	387.48
Formula	C₂₀H₂₉N₅O₃
Cas No.	34661-75-1
Smiles	O(C)C1=C(C=CC=C1)N2CCN(CCCNC=3N(C)C(=O)N(C)C(=O)C3)CC2
Relative Density.	1.2058 g/cm3 (Estimated)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

H2O: < 0.1 mg/mL (insoluble)

DMSO: 50 mg/mL (129.04 mM), Sonication is recommended.

In Vivo Formulation

10% DMSO+40% PEG300+5% Tween 80+45% Saline: 2 mg/mL (5.16 mM), Sonication is recommended.

Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.5808 mL	12.9039 mL	25.8078 mL	129.0389 mL
5 mM	0.5162 mL	2.5808 mL	5.1616 mL	25.8078 mL
10 mM	0.2581 mL	1.2904 mL	2.5808 mL	12.9039 mL
20 mM	0.1290 mL	0.6452 mL	1.2904 mL	6.4519 mL
50 mM	0.0516 mL	0.2581 mL	0.5162 mL	2.5808 mL
100 mM	0.0258 mL	0.1290 mL	0.2581 mL	1.2904 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc