AZD-5991 Racemate

Name: AZD-5991 Racemate
Brand: TargetMol
SKU: T10434L
Price: 139 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T10434LCas No. 2143010-83-5

Alias AZD5991 Racemate, (Rac)-AZD-5991

AZD-5991 Racemate is the racemate of AZD-5991. (Rac)-AZD-5991 is a novel Mcl-1 inhibitor with IC50 <3 nM in FRET assay and induces upregulation of BCL2,BCL-XL, CMYC and MCL1 in AML cell lines.

AZD-5991 Racemate

🥰Excellent

Catalog No. T10434LAlias AZD5991 Racemate, (Rac)-AZD-5991Cas No. 2143010-83-5

AZD-5991 Racemate is the racemate of AZD-5991. (Rac)-AZD-5991 is a novel Mcl-1 inhibitor with IC50 <3 nM in FRET assay and induces upregulation of BCL2,BCL-XL, CMYC and MCL1 in AML cell lines.

Pack Size	Price	Availability
1 mg	$139	In Stock
5 mg	$469	In Stock
10 mg	$687	In Stock

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Product Introduction

Bioactivity

Description	AZD-5991 Racemate is the racemate of AZD-5991. (Rac)-AZD-5991 is a novel Mcl-1 inhibitor with IC50 <3 nM in FRET assay and induces upregulation of BCL2,BCL-XL, CMYC and MCL1 in AML cell lines.
Targets&IC50	MCL1:<3 nM
In vitro	AZD-5991 Racemate is a potent Mcl-1 inhibitor, showing an IC₅₀ below 3 nM in a FRET-based assay[1].
Synonyms	AZD5991 Racemate, (Rac)-AZD-5991

Chemical Properties

Molecular Weight	672.26
Formula	C₃₅H₃₄ClN₅O₃S₂
Cas No.	2143010-83-5
Smiles	O=C(O)C1=C2C=3C=CC(Cl)=C(C=4C(=NN(C4C)C)CSCC5=NN(C(=C5)CSC=6C=C(OCCC2)C=7C=CC=CC7C6)C)C3N1C
Relative Density.	no data available

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store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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