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CDK9-IN-1

Name: CDK9-IN-1
Brand: TargetMol
SKU: T10741
Price: 35 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T10741Cas No. 1415559-43-1

CDK9-IN-1 is a selective and potent CDK9 inhibitor with antiviral activity used in the study of PRRSV infections.

CDK9-IN-1

🥰Excellent

Purity: 98.52%

Catalog No. T10741Cas No. 1415559-43-1

CDK9-IN-1 is a selective and potent CDK9 inhibitor with antiviral activity used in the study of PRRSV infections.

Pack Size	Price	Availability	Quantity
1 mg	$35	In Stock

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Purity:98.52%

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Product Introduction

Bioactivity

Description	CDK9-IN-1 is a selective and potent CDK9 inhibitor with antiviral activity used in the study of PRRSV infections.
Targets&IC50	CDK9-CyclinT1:39 nM
In vitro	CDK9-IN-1 is a selective CDK9 inhibitor with an IC50 = 39 nM for CDK9/CycT1. p24 analysis of CDK9-IN-1 revealed that it can be used for the treatment of HIV infection. [1]

Chemical Properties

Molecular Weight	499.54
Formula	C₂₆H₂₁N₅O₄S
Cas No.	1415559-43-1
Smiles	O=C1C=2C=CC=CC2C(=O)N1C3=CC=CC(=C3)C=4N=CN=C(C4)NC5=CC=C(C(=C5)NS(=O)(=O)C)C
Relative Density.	1.463 g/cm3 (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 80 mg/mL(160.15 mM), Sonication is recommended.

H2O: < 0.1 mg/mL (insoluble)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0018 mL	10.0092 mL	20.0184 mL	100.0921 mL
5 mM	0.4004 mL	2.0018 mL	4.0037 mL	20.0184 mL
10 mM	0.2002 mL	1.0009 mL	2.0018 mL	10.0092 mL
20 mM	0.1001 mL	0.5005 mL	1.0009 mL	5.0046 mL
50 mM	0.0400 mL	0.2002 mL	0.4004 mL	2.0018 mL
100 mM	0.0200 mL	0.1001 mL	0.2002 mL	1.0009 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc