Powder: -20°C for 3 years | In solvent: -80°C for 1 year
AChE/BChE/MAO-B-IN-1 is a reversible, non-time-dependent inhibitor of AChE, BChE and MAO-B that crosses the blood-brain barrier and exhibits inhibitory effects on hAChE, hBChE and hMAO-B with IC50s of 7.31, 0.56 and 26.1 μM, respectively. 1 had a neuroprotective effect and was not significantly cytotoxic.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 195.00 | |
5 mg | In stock | $ 440.00 | |
10 mg | In stock | $ 648.00 | |
25 mg | In stock | $ 987.00 | |
50 mg | In stock | $ 1,390.00 | |
100 mg | In stock | $ 1,870.00 | |
500 mg | In stock | $ 3,730.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 443.00 |
Description | AChE/BChE/MAO-B-IN-1 is a reversible, non-time-dependent inhibitor of AChE, BChE and MAO-B that crosses the blood-brain barrier and exhibits inhibitory effects on hAChE, hBChE and hMAO-B with IC50s of 7.31, 0.56 and 26.1 μM, respectively. 1 had a neuroprotective effect and was not significantly cytotoxic. |
Targets&IC50 | AChE:7.31 μM, BChE:0.56 μM, MAO-B:26.1 μM |
In vitro | AChE/BChE/MAO-B-IN-1 inhibits neuronal cell death induced by amyloid β 1-42 (Aβ 1-42).[1] |
Molecular Weight | 324.42 |
Formula | C20H24N2O2 |
CAS No. | 2416910-82-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 27.5 mg/mL (84.77 mM)
You can also refer to dose conversion for different animals. More
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AChE/BChE/MAO-B-IN-1 2416910-82-0 Metabolism Neuroscience MAO AChE inhibitor inhibit