Powder: -20°C for 3 years | In solvent: -80°C for 1 year
BR102910 (4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]-) is a selective inhibitor of fibroblast activated protein (FAP).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 218.00 | |
5 mg | In stock | $ 553.00 | |
10 mg | In stock | $ 797.00 | |
25 mg | In stock | $ 1,220.00 | |
50 mg | In stock | $ 1,650.00 | |
100 mg | In stock | $ 2,220.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 639.00 |
Description | BR102910 (4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]-) is a selective inhibitor of fibroblast activated protein (FAP). |
In vivo | 4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]-(C57BL/6J mice, 0-30 mg/kg, orally, once) showed significant FAP inhibition in a dose dependent manner [1]. |
Synonyms | 4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]- |
Molecular Weight | 459.3 |
Formula | C18H14Cl2F2N4O2S |
CAS No. | 2505339-54-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 55 mg/mL (119.75 mM)
You can also refer to dose conversion for different animals. More
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BR102910 2505339-54-6 Others FAP Inhibitor POP 4-Thiazolecarboxamide, N-[2-[(2S)-2-cyano-4,4-difluoro-1-pyrrolidinyl]-2-oxoethyl]-2-[(3,4-dichlorophenyl)methyl]- inhibit BR102910 prolyl oligopeptidase BR-102910 Inhibitor Prolyl Endopeptidase (PREP) BR 102910 inhibitor