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idalopirdine

Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.

Catalog No. T7103Cas No. 467459-31-0

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Purity:98%

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idalopirdine

Catalog No. T7103Cas No. 467459-31-0

Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Pack Size	Price	Availability
1 mg	$48	In Stock
5 mg	$119	In Stock
10 mg	$160	In Stock
25 mg	$271	In Stock
50 mg	$398	In Stock
100 mg	$567	In Stock
200 mg	$772	In Stock
1 mL x 10 mM (in DMSO)	$118	In Stock

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Product Introduction

Bioactivity

Description	Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.
Targets&IC50	5-HT6:0.83 nM(Ki)
Alias	Lu AE58054

Chemical Properties

Molecular Weight	398.37
Formula	C₂₀H₁₉F₅N₂O
Cas No.	467459-31-0

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 55 mg/mL (138.06 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.5102 mL	12.5511 mL	25.1023 mL	125.5115 mL
5 mM	0.5020 mL	2.5102 mL	5.0205 mL	25.1023 mL
10 mM	0.2510 mL	1.2551 mL	2.5102 mL	12.5511 mL
20 mM	0.1255 mL	0.6276 mL	1.2551 mL	6.2756 mL
50 mM	0.0502 mL	0.2510 mL	0.5020 mL	2.5102 mL
100 mM	0.0251 mL	0.1255 mL	0.2510 mL	1.2551 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc