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idalopirdine

🥰Excellent
Catalog No. T7103Cas No. 467459-31-0
Alias Lu AE58054

Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.

idalopirdine
Other Forms of idalopirdine:
Idalopirdine HydrochlorideT22936467458-02-2
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idalopirdine

🥰Excellent
Purity: 99.73%
Catalog No. T7103Alias Lu AE58054Cas No. 467459-31-0
Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$81In StockIn Stock
2 mg$121In StockIn Stock
5 mg$198In StockIn Stock
10 mg$267In StockIn Stock
25 mg$451In StockIn Stock
50 mg$663In StockIn Stock
100 mg$945In StockIn Stock
1 mL x 10 mM (in DMSO)$197In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Batch Information

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Purity:99.73%
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Product Introduction

Bioactivity
Description
Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.
Targets&IC50
5-HT6:0.83 nM(Ki)
SynonymsLu AE58054
Chemical Properties
Molecular Weight398.37
FormulaC20H19F5N2O
Cas No.467459-31-0
SmilesC(CNCC1=CC(OCC(C(F)F)(F)F)=CC=C1)C=2C=3C(NC2)=CC(F)=CC3
Relative Density.1.309 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 55 mg/mL (138.06 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.5102 mL12.5511 mL25.1023 mL125.5115 mL
5 mM0.5020 mL2.5102 mL5.0205 mL25.1023 mL
10 mM0.2510 mL1.2551 mL2.5102 mL12.5511 mL
20 mM0.1255 mL0.6276 mL1.2551 mL6.2756 mL
50 mM0.0502 mL0.2510 mL0.5020 mL2.5102 mL
100 mM0.0251 mL0.1255 mL0.2510 mL1.2551 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
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Keywords

Serotonin ReceptorLu AE-58054Lu AE 58054Inhibitorinhibitidalopirdine5-hydroxytryptamine Receptor5HTReceptor5-HT65-HT Receptor5HT Receptor
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