Shopping Cart

Remove All

Your shopping cart is currently empty

Proceed to checkout Continue shopping

Sodium Channel inhibitor 6

Name: Sodium Channel inhibitor 6
Brand: TargetMol
SKU: T204460
Rating: 4.5 (1 reviews)

😃Good

Catalog No. T204460Cas No. 2877755-11-6

Sodium Channel inhibitor 6 (Compound I) is an effective sodium channel antagonist for neuropathic pain research.

Sodium Channel inhibitor 6

😃Good

Catalog No. T204460Cas No. 2877755-11-6

Sodium Channel inhibitor 6 (Compound I) is an effective sodium channel antagonist for neuropathic pain research.

Pack Size	Price	USA Warehouse	Global Warehouse	Quantity
10 mg	Inquiry	10-14 weeks	10-14 weeks
50 mg	Inquiry	10-14 weeks	10-14 weeks

Add to Quotation

In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

Select Batch

Resource Download

COA

Product Introduction

Bioactivity

Description

Sodium Channel inhibitor 6 (Compound I) is an effective sodium channel antagonist for neuropathic pain research.

Chemical Properties

Molecular Weight	490.42
Formula	C₂₂H₂₃F₅N₂O₅
Cas No.	2877755-11-6
Smiles	C(NC=1C=CC([C@H](CO)O)=NC1)(=O)[C@H]2[C@@H]([C@H](C)[C@@](C(F)(F)F)(C)O2)C3=C(OC)C(F)=C(F)C=C3
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 200 mg/mL (407.81 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0391 mL	10.1953 mL	20.3907 mL	101.9534 mL
5 mM	0.4078 mL	2.0391 mL	4.0781 mL	20.3907 mL
10 mM	0.2039 mL	1.0195 mL	2.0391 mL	10.1953 mL
20 mM	0.1020 mL	0.5098 mL	1.0195 mL	5.0977 mL
50 mM	0.0408 mL	0.2039 mL	0.4078 mL	2.0391 mL
100 mM	0.0204 mL	0.1020 mL	0.2039 mL	1.0195 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline /PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline /PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc