Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Steroid sulfatase-IN-1 is a highly potent and orally active inhibitor of the enzyme Steroid sulfatase, with an impressive IC50 value of 1.71 μM. This compound exhibits notable antitumor activity, achieving a TGI (tumor growth inhibition) of 51% in vivo. Therefore, Steroid sulfatase-IN-1 holds great promise in the field of breast cancer research [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | Steroid sulfatase-IN-1 is a highly potent and orally active inhibitor of the enzyme Steroid sulfatase, with an impressive IC50 value of 1.71 μM. This compound exhibits notable antitumor activity, achieving a TGI (tumor growth inhibition) of 51% in vivo. Therefore, Steroid sulfatase-IN-1 holds great promise in the field of breast cancer research [1]. |
In vivo | Steroid sulfatase-IN-1 (compound 4 b), administered orally at a dosage of 50 mg/kg, demonstrates notable antitumor efficacy, achieving a tumor growth inhibition (TGI) value of 51% in a 67NR mouse model. |
Molecular Weight | 385.23 |
Formula | C14H10Cl2N4O3S |
CAS No. | 2403716-19-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Steroid sulfatase-IN-1 2403716-19-6 inhibitor inhibit