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(Rac)-Pyrotinib

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Catalog No. T38633Cas No. 1246089-97-3
Alias (Rac)-SHR-1258, (Rac)-Pyrotinib

(Rac)-Pyrotinib ((Rac)-SHR-1258) is the racemate of Pyrotinib, a potent and selective EGFR/HER2 dual inhibitor.

(Rac)-Pyrotinib
Other Forms of (Rac)-Pyrotinib:
Pyrotinib dimaleateT125941397922-61-0
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(Rac)-Pyrotinib

🥰Excellent
Catalog No. T38633Alias (Rac)-SHR-1258, (Rac)-PyrotinibCas No. 1246089-97-3
(Rac)-Pyrotinib ((Rac)-SHR-1258) is the racemate of Pyrotinib, a potent and selective EGFR/HER2 dual inhibitor.
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Product Introduction

Bioactivity
Description
(Rac)-Pyrotinib ((Rac)-SHR-1258) is the racemate of Pyrotinib, a potent and selective EGFR/HER2 dual inhibitor.
Synonyms(Rac)-SHR-1258, (Rac)-Pyrotinib
Chemical Properties
Molecular Weight583.09
FormulaC32H31ClN6O3
Cas No.1246089-97-3
SmilesCCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\C1CCCN1C
Relative Density.1.35 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
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Keywords

SHR-1258SHR1258SHR 1258Pyrotinib(Rac)Pyrotinib(Rac) Pyrotinib
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