Powder: -20°C for 3 years | In solvent: -80°C for 1 year
YAP-TEAD-IN-3 is an inhibitor of YAP/TAZ-TEAD interactions with an IC50 of 9 nM for Avi-human TEAD (4217-434). YAP-TEAD-IN-3 inhibits YAP reporter gene expression (IC50 = 0.048 μM) and NCI-H2052 cell proliferation (IC50 = 0.048 μM).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | Inquiry | $ 328.00 | |
5 mg | Inquiry | $ 783.00 | |
10 mg | Inquiry | $ 1,060.00 | |
25 mg | Inquiry | $ 1,580.00 | |
50 mg | Inquiry | $ 2,130.00 | |
100 mg | Inquiry | $ 2,880.00 |
Description | YAP-TEAD-IN-3 is an inhibitor of YAP/TAZ-TEAD interactions with an IC50 of 9 nM for Avi-human TEAD (4217-434). YAP-TEAD-IN-3 inhibits YAP reporter gene expression (IC50 = 0.048 μM) and NCI-H2052 cell proliferation (IC50 = 0.048 μM). |
Targets&IC50 | YAP-TEAD:9 nM |
Synonyms | IAG933 |
Molecular Weight | 529.96 |
Formula | C27H26ClF2N3O4 |
CAS No. | 2714434-21-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (94.34 mM), Sonication is recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
YAP-TEAD-IN-3 2714434-21-4 Stem Cells YAP YAPTEADIN3 IAG933 inhibitor inhibit